SCHEMBL8489654

SCHEMBL8489654

CCCCCCCCN(CC(O)C[Gd]N1CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC1)S(C)(=O)=O

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.36
PER2 O15055 3/20 0.33
CRY1 Q16526 2/20 0.31
CRY2 Q49AN0 2/20 0.31
GPR84 Q9NQS5 4/20 0.30
SIGMAR1 Q99720 1/20 0.30
MMP1 P03956 1/20 0.30
MMP2 P08253 1/20 0.30
MMP3 P08254 1/20 0.30
MMP8 P22894 1/20 0.30
MMP13 P45452 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8486390 1.00 S1PR1 (0.36) S1PR1PER2CRY1CRY2GPR84
SCHEMBL8488567 0.96 PER2 (0.34) S1PR1PER2CRY1CRY2SIGMAR1
SCHEMBL8490612 0.85 PER2 (0.40) S1PR1PER2CRY1CRY2
SCHEMBL8485649 0.85 PER2 (0.40) S1PR1PER2CRY1CRY2
SCHEMBL8488046 0.85 PER2 (0.42) PER2CRY1CRY2
SCHEMBL8488408 0.81 PER2 (0.51) PER2CRY1CRY2
SCHEMBL8489932 0.80 PER2 (0.42) S1PR1PER2CRY1CRY2
SCHEMBL8484814 0.79 CRY1 (0.49) PER2CRY1CRY2
SCHEMBL8486007 0.78 LMNA (0.44) PER2CRY1CRY2
SCHEMBL8487214 0.72 PER2 (0.38) PER2CRY1CRY2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919431-A 1,4,7,10-tetraazacyclododecane derivatives, their use, pharmaceutical agents containing these compounds and process for their production SCHERING AKTIENGESELLSCHAFT (DE) 1999-07-06 US disclosed