SCHEMBL8486004

SCHEMBL8486004

Oc1ccc(C(Cc2ccccc2)CC(O)C2(O)CCNCC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.39
ESR2 Q92731 3/20 0.39
ADRA1A P35348 3/20 0.39
GRIN2B Q13224 3/20 0.39
ADRA1D P25100 2/20 0.39
ADRA1B P35368 2/20 0.39
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2C Q14957 1/20 0.39
GRIN3A Q8TCU5 1/20 0.39
SLC6A2 P23975 2/20 0.36
LMNA P02545 1/20 0.36
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8486958 0.99 ESR1 (0.38) ESR1ESR2ADRA1AGRIN2BADRA1D
SCHEMBL8482269 0.88 GRIN2D (0.41) ESR1ESR2ADRA1AGRIN2BADRA1D
SCHEMBL8487882 0.80 GRIN2D (0.37) ADRA1AGRIN2BADRA1DADRA1BGRIN2D
Hydrochloric Acid SCHEMBL8482025 0.79 GRIN2D (0.36) ADRA1AGRIN2BADRA1DADRA1BGRIN2D
SCHEMBL27564167 0.72 ESR1 (0.62) ESR1ESR2SLC6A2LMNASLC6A3
SCHEMBL8570543 0.69 EPHX1 (0.42) SLC6A2OPRM1SLC6A3CYP2D6TSHR
SCHEMBL5374718 0.68 RAB9A (0.41) ADRB2
SCHEMBL15288809 0.68 ESR1 (0.56) ESR1ESR2CYP1A2CYP3A4CYP2C19
SCHEMBL15288808 0.68 ESR1 (0.56) ESR1ESR2CYP1A2CYP3A4CYP2C19
SCHEMBL9498596 0.68 ESR1 (0.60) ESR1ESR2SLC6A2TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889026-A 4-hydroxy-piperodine derivatives HOFFMANN-LA ROCHE INC. (US) 1999-03-30 US disclosed