SCHEMBL8486953

SCHEMBL8486953

CS(=O)(=O)NC(C(O)CN1CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC1)C1COC(c2ccccc2)OC1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 1/20 0.37
KDM1A O60341 4/20 0.36
MOGAT2 Q3SYC2 2/20 0.36
ADRB2 P07550 4/20 0.34
ADRB1 P08588 4/20 0.34
ADRB3 P13945 4/20 0.34
SLC18A3 Q16572 2/20 0.34
PRCP P42785 1/20 0.31
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA7 P43166 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8489440 0.89 HCRTR2 (0.37) HCRTR2MOGAT2ADRB2ADRB1ADRB3
SCHEMBL9004363 0.74 PER2 (0.52)
SCHEMBL8491337 0.67 TSHR (0.39) ADRB2ADRB1ADRB3CA1CA2
SCHEMBL27648542 0.63 MEN1 (0.50) SLC18A3
SCHEMBL23816922 0.62 SLC18A3 (0.60) SLC18A3
SCHEMBL8489489 0.62 CRY1 (0.60)
SCHEMBL7202138 0.61 SLC18A3 (0.62) SLC18A3
SCHEMBL13377720 0.61 MEN1 (0.36) HCRTR2MOGAT2
SCHEMBL13377724 0.59 TSHR (0.46)
SCHEMBL13381275 0.59 MEN1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919431-A 1,4,7,10-tetraazacyclododecane derivatives, their use, pharmaceutical agents containing these compounds and process for their production SCHERING AKTIENGESELLSCHAFT (DE) 1999-07-06 US disclosed