SCHEMBL9004363

SCHEMBL9004363

CS(=O)(=O)N(CC(O)CN1CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC1)C1COC(c2ccccc2)OC1

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PER2 O15055 20/20 0.52
CRY1 Q16526 18/20 0.47
CRY2 Q49AN0 18/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9004331 0.89 PER2 (0.47) PER2CRY1CRY2
SCHEMBL8489489 0.75 CRY1 (0.60) PER2CRY1CRY2
SCHEMBL8486953 0.74 HCRTR2 (0.37)
SCHEMBL9004352 0.71 PER2 (0.43) PER2CRY1CRY2
SCHEMBL9004320 0.69 PER2 (0.46) PER2CRY1CRY2
SCHEMBL9004350 0.69 MAPT (0.37) PER2CRY1CRY2
SCHEMBL9004290 0.68 PER2 (0.38) PER2CRY1CRY2
SCHEMBL8489932 0.67 PER2 (0.42) PER2CRY1CRY2
SCHEMBL5557205 0.67 ALDH1A1 (0.46)
SCHEMBL8485649 0.66 PER2 (0.40) PER2CRY1CRY2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730586-A1 1,4,7,10-TETRAAZACYCLODODECANE DERIVATIVES, THEIR USE, PHARMACEUTICALS CONTAINING THEM AND PROCESS FOR THEIR PRODUCTION SCHERING AKTIENGESELLSCHAFT (DE) 1996-09-11 EP disclosed
WO-1995014678-A1 1,4,7,10-TETRAAZACYCLODODECANE DERIVATIVES, THEIR USE, PHARMACEUTICALS CONTAINING THEM AND PROCESS FOR THEIR PRODUCTION SCHERING AKTIENGESELLSCHAFT (DE) 1995-06-01 WO disclosed