SCHEMBL8489489

SCHEMBL8489489

CS(=O)(=O)N(Cc1ccccc1)CC(O)CN1CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CRY1 Q16526 7/20 0.60
CRY2 Q49AN0 7/20 0.60
PER2 O15055 6/20 0.60
BACE1 P56817 8/20 0.53
SMN1; SMN2 Q16637 2/20 0.44
ALDH1A1 P00352 2/20 0.44
POLB P06746 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8487228 0.87 CRY1 (0.53) CRY1CRY2PER2BACE1SMN1; SMN2
SCHEMBL8484814 0.86 CRY1 (0.49) CRY1CRY2PER2BACE1SMN1; SMN2
SCHEMBL9004320 0.84 PER2 (0.46) CRY1CRY2PER2BACE1ALDH1A1
SCHEMBL5557205 0.83 ALDH1A1 (0.46) BACE1SMN1; SMN2ALDH1A1POLBMEN1
SCHEMBL9004350 0.80 MAPT (0.37) CRY1CRY2PER2BACE1KMT2A
SCHEMBL18975189 0.80 ALDH1A1 (0.44) BACE1SMN1; SMN2ALDH1A1POLBMEN1
SCHEMBL9004290 0.79 PER2 (0.38) CRY1CRY2PER2BACE1KMT2A
SCHEMBL8489932 0.78 PER2 (0.42) CRY1CRY2PER2BACE1ALDH1A1
SCHEMBL8488572 0.78 BACE1 (0.48) CRY1CRY2PER2BACE1ALDH1A1
SCHEMBL8489557 0.77 PER2 (0.55) CRY1CRY2PER2BACE1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919431-A 1,4,7,10-tetraazacyclododecane derivatives, their use, pharmaceutical agents containing these compounds and process for their production SCHERING AKTIENGESELLSCHAFT (DE) 1999-07-06 US disclosed
EP-0730586-A1 1,4,7,10-TETRAAZACYCLODODECANE DERIVATIVES, THEIR USE, PHARMACEUTICALS CONTAINING THEM AND PROCESS FOR THEIR PRODUCTION SCHERING AKTIENGESELLSCHAFT (DE) 1996-09-11 EP disclosed
WO-1995014678-A1 1,4,7,10-TETRAAZACYCLODODECANE DERIVATIVES, THEIR USE, PHARMACEUTICALS CONTAINING THEM AND PROCESS FOR THEIR PRODUCTION SCHERING AKTIENGESELLSCHAFT (DE) 1995-06-01 WO disclosed