SCHEMBL8486969

SCHEMBL8486969

CN1C(=O)C(=Cc2ccccc2)c2cc(-c3csc(-c4ccncc4)n3)ccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.46
AR P10275 2/20 0.46
KMT2A Q03164 2/20 0.46
SMN1; SMN2 Q16637 4/20 0.42
RAB9A P51151 3/20 0.42
NPC1 O15118 2/20 0.42
LMNA P02545 2/20 0.42
BCL2 P10415 2/20 0.41
BAX Q07812 2/20 0.41
BCL2L1 Q07817 2/20 0.41
CDK5 Q00535 2/20 0.41
CDK5R1 Q15078 2/20 0.41
CYP19A1 P11511 4/20 0.41
MAPT P10636 3/20 0.41
POLB P06746 2/20 0.41
STAT3 P40763 1/20 0.41
ERBB2 P04626 1/20 0.41
CDC25A P30304 1/20 0.41
CDC25B P30305 1/20 0.41
CDC25C P30307 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8483385 0.85 KDM4E (0.45) KDM4EARKMT2ASMN1; SMN2RAB9A
SCHEMBL8479782 0.84 KDM4E (0.43) KDM4EARKMT2ASMN1; SMN2RAB9A
SCHEMBL8484634 0.82 KDM4E (0.50) KDM4EARKMT2ASMN1; SMN2RAB9A
SCHEMBL8480783 0.76 CYP19A1 (0.46) KDM4EARKMT2ASMN1; SMN2RAB9A
SCHEMBL17875110 0.72 MET (0.44) KMT2ACDK5CDK5R1CDC25ACDC25B
SCHEMBL8486372 0.71 CDC25A (0.72) KDM4EARKMT2ASMN1; SMN2RAB9A
SCHEMBL8485576 0.70 KDM4E (0.47) KDM4EARKMT2ASMN1; SMN2RAB9A
SCHEMBL8524349 0.70 CDC25A (0.59) KDM4EARSMN1; SMN2RAB9ANPC1
SCHEMBL8524907 0.70 KDM4E (0.49) KDM4EARKMT2ASMN1; SMN2RAB9A
SCHEMBL8484951 0.69 KDM4E (0.48) KDM4EARKMT2ASMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999015524-A1 THIAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-04-01 WO disclosed