SCHEMBL8488579

SCHEMBL8488579

COc1ccc(CCN(C2CN(CC(C)O)CCN(CC(=O)O)CCN(CC(=O)O)CCN2CC(=O)O)S(C)(=O)=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.39
CCR5 P51681 3/20 0.37
ALDH1A1 P00352 3/20 0.36
SLC6A9 P48067 2/20 0.35
CHRM5 P08912 3/20 0.35
CHRM1 P11229 3/20 0.35
CHRM3 P20309 3/20 0.35
SIGMAR1 Q99720 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
ALOX5 P09917 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
POLB P06746 1/20 0.35
RAB9A P51151 1/20 0.35
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8488757 0.82 PER2 (0.30)
SCHEMBL8489492 0.81 MAPK1 (0.40) LMNAALDH1A1SLC6A9POLB
SCHEMBL8488416 0.81 ALDH1A1 (0.39) LMNAALDH1A1SMN1; SMN2POLBBACE1
SCHEMBL8489560 0.80 ALDH1A1 (0.37) ALDH1A1SMN1; SMN2POLB
SCHEMBL8489937 0.80 SIGMAR1 (0.33) SIGMAR1
SCHEMBL8490617 0.78 S1PR1 (0.36) SIGMAR1
SCHEMBL8485655 0.78 S1PR1 (0.36) SIGMAR1
SCHEMBL8488572 0.76 BACE1 (0.48) LMNAALDH1A1BACE1
SCHEMBL8488562 0.73 ALDH1A1 (0.35) LMNAALDH1A1CHRM5CHRM1CHRM3
SCHEMBL8488054 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919431-A 1,4,7,10-tetraazacyclododecane derivatives, their use, pharmaceutical agents containing these compounds and process for their production SCHERING AKTIENGESELLSCHAFT (DE) 1999-07-06 US disclosed