SCHEMBL8488562

SCHEMBL8488562

COc1ccc(CCN(C2C(CCCO)NCCN(CC(=O)O)CCN(CC(=O)O)CCN2CC(=O)O)S(C)(=O)=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
CHRM5 P08912 4/20 0.35
CHRM1 P11229 4/20 0.35
CHRM3 P20309 4/20 0.35
SIGMAR1 Q99720 2/20 0.34
OPRM1 P35372 2/20 0.33
C5AR1 P21730 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
DRD2 P14416 1/20 0.33
MMP1 P03956 1/20 0.33
MMP9 P14780 1/20 0.33
MMP13 P45452 1/20 0.33
ADAM17 P78536 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8487892 0.89 SIGMAR1 (0.34) ALDH1A1LMNACHRM5CHRM1CHRM3
SCHEMBL8488750 0.84
SCHEMBL8489481 0.82 MAPK1 (0.35) ALDH1A1LMNASIGMAR1
SCHEMBL8489922 0.82 SIGMAR1 (0.33) SIGMAR1
SCHEMBL8488579 0.73 LMNA (0.39) ALDH1A1LMNACHRM5CHRM1CHRM3
SCHEMBL8491774 0.73
SCHEMBL8488572 0.68 BACE1 (0.48) ALDH1A1LMNA
SCHEMBL8486007 0.65 LMNA (0.44) ALDH1A1LMNACHRM5CHRM1CHRM3
SCHEMBL8482567 0.61 ITGB3 (0.40) ALDH1A1
SCHEMBL8482371 0.61 DRD2 (0.41) ALDH1A1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919431-A 1,4,7,10-tetraazacyclododecane derivatives, their use, pharmaceutical agents containing these compounds and process for their production SCHERING AKTIENGESELLSCHAFT (DE) 1999-07-06 US disclosed