SCHEMBL8489385

SCHEMBL8489385

C=CC(=O)Oc1cc2c(Nc3ccc(OCc4ccccc4)cc3)ncnc2cc1OCCCCN(C)C

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.57
ERBB2 P04626 10/20 0.57
ERBB4 Q15303 2/20 0.53
CHEK2 O96017 1/20 0.48
ROS1 P08922 1/20 0.48
FLT3 P36888 1/20 0.48
AURKB Q96GD4 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48
MKNK2 Q9HBH9 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8486258 0.91 EGFR (0.60) EGFRERBB2ERBB4AURKB
SCHEMBL7243958 0.87 EGFR (0.71) EGFRERBB2ERBB4
SCHEMBL7235690 0.85 EGFR (0.55) EGFRERBB2ERBB4CHEK2ROS1
SCHEMBL7235693 0.84 EGFR (0.54) EGFRERBB2ERBB4CHEK2ROS1
SCHEMBL8525841 0.83 EGFR (0.61) EGFRERBB2ERBB4FLT3AURKB
SCHEMBL8154615 0.81 EGFR (0.77) EGFRERBB2ERBB4CHEK2ROS1
SCHEMBL8143063 0.81 EGFR (0.68) EGFRERBB2ERBB4CHEK2ROS1
SCHEMBL28523377 0.81 EGFR (0.51) EGFR
SCHEMBL8490274 0.80 EGFR (0.54) EGFRERBB2
SCHEMBL8809158 0.80 EGFR (0.67) EGFRERBB2ERBB4CHEK2ROS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999006378-A1 IRREVERSIBLE INHIBITORS OF TYROSINE KINASES WARNER-LAMBERT COMPANY (US) 1999-02-11 WO disclosed