SCHEMBL8489557

SCHEMBL8489557

CCOC(=O)CN1CCN(CC(=O)OCC)CCN(CC(O)CN(CCc2ccccc2)S(C)(=O)=O)CCN(CC(=O)OCC)CC1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PER2 O15055 4/20 0.55
CRY1 Q16526 3/20 0.55
CRY2 Q49AN0 3/20 0.55
BACE1 P56817 7/20 0.53
TSHR P16473 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
ALDH1A1 P00352 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ALOX15 P16050 1/20 0.42
CASP1 P29466 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8487228 0.90 CRY1 (0.53) PER2CRY1CRY2BACE1ALDH1A1
SCHEMBL8487896 0.90 BACE1 (0.44) PER2CRY1CRY2BACE1ALDH1A1
SCHEMBL9004296 0.89 PER2 (0.43) PER2CRY1CRY2BACE1TSHR
SCHEMBL8491767 0.83 PER2 (0.39) PER2CRY1CRY2ALDH1A1L3MBTL1
SCHEMBL8488600 0.81 PER2 (0.38) PER2CRY1CRY2ALDH1A1L3MBTL1
SCHEMBL8491775 0.81 PER2 (0.47) PER2CRY1CRY2ALDH1A1L3MBTL1
SCHEMBL8487214 0.81 PER2 (0.38) PER2CRY1CRY2ALDH1A1L3MBTL1
SCHEMBL8488572 0.79 BACE1 (0.48) PER2CRY1CRY2BACE1ALDH1A1
SCHEMBL9004320 0.77 PER2 (0.46) PER2CRY1CRY2BACE1TSHR
SCHEMBL8489489 0.77 CRY1 (0.60) PER2CRY1CRY2BACE1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919431-A 1,4,7,10-tetraazacyclododecane derivatives, their use, pharmaceutical agents containing these compounds and process for their production SCHERING AKTIENGESELLSCHAFT (DE) 1999-07-06 US disclosed
EP-0730586-A1 1,4,7,10-TETRAAZACYCLODODECANE DERIVATIVES, THEIR USE, PHARMACEUTICALS CONTAINING THEM AND PROCESS FOR THEIR PRODUCTION SCHERING AKTIENGESELLSCHAFT (DE) 1996-09-11 EP disclosed
WO-1995014678-A1 1,4,7,10-TETRAAZACYCLODODECANE DERIVATIVES, THEIR USE, PHARMACEUTICALS CONTAINING THEM AND PROCESS FOR THEIR PRODUCTION SCHERING AKTIENGESELLSCHAFT (DE) 1995-06-01 WO disclosed