SCHEMBL8491963

SCHEMBL8491963

N[C@@H](CCc1ccccc1)C(=O)O[C@H](CCCCN1C(=O)c2ccccc2C1=O)C(=O)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
HDAC1 Q13547 3/20 0.43
HDAC7 Q8WUI4 3/20 0.43
CASP3 P42574 1/20 0.43
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
ACHE P22303 4/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Leucine SCHEMBL8488907 0.84 ELANE (0.44) L3MBTL1TDP1HDAC1HDAC7CASP3
SCHEMBL7329031 0.76 TDP1 (0.49) L3MBTL1TDP1HDAC1HDAC7CASP3
SCHEMBL6578347 0.75 TDP1 (0.51) L3MBTL1TDP1HDAC1HDAC7CASP3
Leucine SCHEMBL8524451 0.74 MMP1 (0.47) L3MBTL1TDP1
SCHEMBL8966420 0.74 ALDH1A1 (0.50) L3MBTL1TDP1MAPK1ALDH1A1
SCHEMBL5019164 0.74 ALDH1A1 (0.50) L3MBTL1TDP1MAPK1ALDH1A1
SCHEMBL1245400 0.74 ALDH1A1 (0.50) L3MBTL1TDP1MAPK1ALDH1A1
SCHEMBL408911 0.73 TDP1 (0.49) L3MBTL1TDP1HDAC1HDAC7CASP3
Hydrochloric Acid SCHEMBL29131620 0.73 ALDH1A1 (0.49) L3MBTL1TDP1MAPK1ALDH1A1
Hydrochloric Acid SCHEMBL14119382 0.73 ALDH1A1 (0.49) L3MBTL1TDP1MAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5932551-A INHIBITORS OF MATRIX METALLOENDOPROTEINASE-MEDIATED DISEASES MERCK & CO., INC. (US) 1999-08-03 US disclosed