SCHEMBL8495754

SCHEMBL8495754

CC(C)(C)C.Cc1ccc(NS(=O)(=O)CC2CCCCO2)c(=O)n1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.39
HTT P42858 1/20 0.39
F2 P00734 4/20 0.37
PRSS1 P07477 3/20 0.37
KMO O15229 1/20 0.37
RAB9A P51151 2/20 0.36
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
RCE1 Q9Y256 1/20 0.36
ALDH1A1 P00352 3/20 0.36
ALOX12 P18054 1/20 0.36
MEN1 O00255 2/20 0.36
GAA P10253 2/20 0.36
KMT2A Q03164 2/20 0.36
F10 P00742 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Morpholine SCHEMBL7318127 0.75 F2 (0.35) F2PRSS1F10
SCHEMBL7311770 0.69 F2 (0.34) HTTF2PRSS1ALDH1A1GAA
SCHEMBL16253665 0.65 KMO (0.42) TSHRHTTKMORAB9ALMNA
SCHEMBL7407793 0.64 TSHR (0.36) TSHRHTTKMOSMN1; SMN2MEN1
SCHEMBL23409789 0.61 PKM (0.46) TSHRRAB9AHPGDSMN1; SMN2ALDH1A1
SCHEMBL5070898 0.60 ALDH1A1 (0.50) TSHRHTTMAPTLMNAHPGD
SCHEMBL7322304 0.59 NPC1 (0.55) F2PRSS1RAB9APOLBSMN1; SMN2
SCHEMBL11005143 0.59 GSTO1 (0.49) TSHRHTTRAB9AMAPTLMNA
SCHEMBL12155310 0.58 ALDH1A1 (0.38) TSHRHTTRAB9AMAPTSMN1; SMN2
SCHEMBL5490567 0.58 HPGD (0.38) HTTRAB9ALMNAPOLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5932606-A Pyrazinone, pyridinone, piperidine and pyrrolidine thrombin inhibitors MERCK & CO., INC. (US) 1999-08-03 US disclosed