SCHEMBL8498201

SCHEMBL8498201

NC(=O)C(C1CN(c2ccccc2)CCN1C(N)=O)[C@H](N)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 3/20 0.43
NOTUM Q6P988 1/20 0.40
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
TSHR P16473 2/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
TP53 P04637 1/20 0.34
FAAH O00519 2/20 0.34
SLC6A9 P48067 1/20 0.34
OPRK1 P41145 1/20 0.34
MAPK1 P28482 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
AKR1C3 P42330 1/20 0.33
SCD5 Q86SK9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3669556 0.94 AGTR2 (0.44) AGTR2NOTUMMEN1KMT2ATSHR
SCHEMBL8192461 0.83 AGTR2 (0.37) AGTR2MEN1KMT2ATSHRALDH1A1
SCHEMBL8592475 0.83 NOTUM (0.44) NOTUMMEN1KMT2ATSHRUSP2
SCHEMBL8592708 0.83 NOTUM (0.44) AGTR2NOTUMMEN1KMT2AALDH1A1
SCHEMBL3447709 0.82 HTR1A (0.50) NOTUMMEN1KMT2ATSHRALDH1A1
SCHEMBL8493524 0.82 DRD2 (0.43) MEN1KMT2ATSHRALDH1A1LMNA
SCHEMBL8984626 0.82 NOTUM (0.48) AGTR2NOTUMMEN1KMT2AALDH1A1
SCHEMBL8984815 0.81 AR (0.39) TSHRALDH1A1LMNAMAPTAKR1C3
SCHEMBL8594519 0.80 KMT2A (0.43) MEN1KMT2AALDH1A1FAAHMAPK1
SCHEMBL8984615 0.80 SLC6A9 (0.46) MEN1KMT2AALDH1A1FAAHSLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655463-B1 Cyclic hexapeptides having endothelin antagonistic activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-09-01 EP claimed
EP-0552417-B1 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-07-07 EP claimed
EP-0528312-B1 Cyclic peptides and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-07-16 EP claimed