SCHEMBL8499335

SCHEMBL8499335

CC1(C)CCSc2ccc(C#COC(=O)c3cccnc3)cc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 10/20 0.57
RARB P10826 10/20 0.57
RARG P13631 10/20 0.57
KMT2A Q03164 4/20 0.57
CYP3A4 P08684 3/20 0.57
CYP26A1 O43174 2/20 0.54
RXRA P19793 2/20 0.39
ALDH1A1 P00352 2/20 0.39
CRABP2 P29373 1/20 0.36
LMNA P02545 3/20 0.35
L3MBTL1 Q9Y468 3/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9765059 0.87 RARB (0.57) RARARARBRARGKMT2ACYP3A4
Tazarotene SCHEMBL995895 0.80 RARB (0.81) RARARARBRARGKMT2ACYP3A4
Tazarotene SCHEMBL28326300 0.79 RARA (0.80) RARARARBRARGKMT2ACYP3A4
SCHEMBL181635 0.76 CYP3A4 (0.52) RARARARBRARGKMT2ACYP3A4
SCHEMBL12371728 0.76 RARB (0.78) RARARARBRARGKMT2ACYP3A4
SCHEMBL9817871 0.74 RARA (0.71) RARARARBRARGKMT2ACYP3A4
SCHEMBL19560666 0.74 RARA (0.82) RARARARBRARGKMT2ACYP3A4
SCHEMBL16913398 0.74 RARB (0.56) RARARARBRARGKMT2ACYP3A4
SCHEMBL19034088 0.73 RARB (0.62) RARARARBRARGKMT2ACYP3A4
SCHEMBL17885756 0.73 RARB (0.81) RARARARBRARGKMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5914334-A A GEL FOR TOPICAL TREATMENT OF BOTH ACNE AND PSORIASIS COMPRISES ETHYL-6(2-(4,4-DIMETHYLTHIOCHROMAN-6-YL)-ETHYNYL) NICOTINATE IN A CARRIER SUCH AS: WATER, EDETATE DISODIUM, POLOXOMERS, HEXYLENE GLYCOL, TROMETHANE, POLYSORBATES ETC. ALLERGAN, INC. (US) 1999-06-22 US claimed
US-5824685-A VISION DEFECTS AND GENE EXPRESSION THE JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE (US) 1998-10-20 US claimed
US-5914334-A A GEL FOR TOPICAL TREATMENT OF BOTH ACNE AND PSORIASIS COMPRISES ETHYL-6(2-(4,4-DIMETHYLTHIOCHROMAN-6-YL)-ETHYNYL) NICOTINATE IN A CARRIER SUCH AS: WATER, EDETATE DISODIUM, POLOXOMERS, HEXYLENE GLYCOL, TROMETHANE, POLYSORBATES ETC. ALLERGAN, INC. (US) 1999-06-22 US disclosed