SCHEMBL8499394

SCHEMBL8499394

COC=CCCc1ccc(CC(=O)O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
HPGD P15428 1/20 0.50
HSD17B10 Q99714 1/20 0.50
CA2 P00918 1/20 0.44
CAMK2A Q9UQM7 1/20 0.44
AKR1B1 P15121 1/20 0.42
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 3/20 0.42
TSHR P16473 2/20 0.42
PTGS1 P23219 2/20 0.42
ABCC4 O15439 1/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
NFKB1 P19838 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
GPR52 Q9Y2T5 5/20 0.41
CYP4F2 P78329 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8499393 1.00 ALDH1A1 (0.50) ALDH1A1HPGDHSD17B10CA2CAMK2A
SCHEMBL5085202 0.78 GPR52 (0.47) GPR52
SCHEMBL23188649 0.77 CYP1A2 (0.43) GPR52
SCHEMBL31422448 0.76 PTGS1 (0.47) ALDH1A1HPGDHSD17B10CA2CAMK2A
SCHEMBL755404 0.75 TAAR1 (0.42) ALDH1A1KDM4EPOLBPTGS1
SCHEMBL755405 0.75 TAAR1 (0.42) ALDH1A1KDM4EPOLBPTGS1
SCHEMBL8503304 0.74 ALDH1A1 (0.55) ALDH1A1HPGDHSD17B10CA2CAMK2A
SCHEMBL9089148 0.74 CYP4A11 (0.41) ALDH1A1HPGDHSD17B10CA2GPR52
SCHEMBL9089152 0.74 CYP4A11 (0.41) ALDH1A1HPGDHSD17B10CA2GPR52
SCHEMBL2996429 0.73 CA2 (0.68) ALDH1A1HPGDHSD17B10CA2CAMK2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5892034-A Process for preparing 5-substituted pyrrolo- 2,3-d!pyrimidines ELI LILLY AND COMPANY (US) 1999-04-06 US disclosed
US-5663339-A Process for preparing 5-substituted pyrrolo-[2,3-D] pyrimidines ELI LILLY AND COMPANY (US) 1997-09-02 US disclosed
US-5644058-A Process for preparing 5-substituted pyrrolo-[2,3-d]pyrimidines ELI LILLY AND COMPANY (US) 1997-07-01 US disclosed
US-5612482-A Process for preparing 5-substituted pyrrolo-[2,3-d]pyrimidines ELI LILLY AND COMPANY (US) 1997-03-18 US disclosed
US-5416211-A Process for preparing 5-substituted pyrrolo-[2,3-d]pyrimidines ELI LILLY AND COMPANY (US) 1995-05-16 US disclosed
EP-0589720-A2 Process for preparing 5-substituted pyrrolo-[2,3-d]pyrimidines ELI LILLY AND COMPANY (US) 1994-03-30 EP disclosed