SCHEMBL8499490

SCHEMBL8499490

OCc1ccc2ccc(F)cc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
CYP2A6 P11509 1/20 0.48
CYP19A1 P11511 1/20 0.47
CA2 P00918 2/20 0.43
CA12 O43570 1/20 0.43
CA3 P07451 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
CA5A P35218 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
CA5B Q9Y2D0 1/20 0.43
SLC6A2 P23975 3/20 0.40
SLC6A4 P31645 3/20 0.40
SLC6A3 Q01959 2/20 0.40
KCNH2 Q12809 2/20 0.40
DAO P14920 2/20 0.38
PTGS1 P23219 1/20 0.37
CYP4F2 P78329 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3517975 0.93 CYP1A2 (0.50) CYP1A2CYP2A6CYP19A1CA2CA12
SCHEMBL3039135 0.86 CA2 (0.52) CYP1A2CYP2A6CA2CA12CA3
SCHEMBL8499350 0.83 KDM4E (0.45) CYP1A2CYP2A6CYP19A1CA2SLC6A2
SCHEMBL13525455 0.79 CA2 (0.50) CYP1A2CYP2A6CA2CA12CA3
SCHEMBL29617406 0.79 CA2 (0.50) CYP1A2CYP2A6CA2CA12CA3
SCHEMBL6959233 0.78 CYP1A2 (0.48) CYP1A2CYP2A6CYP19A1SLC6A2SLC6A4
SCHEMBL14604942 0.78 CYP1A2 (0.59) CYP1A2CYP2A6CYP19A1SLC6A2SLC6A4
SCHEMBL8499487 0.78 CYP1A2 (0.48) CYP1A2CYP2A6CYP19A1SLC6A2SLC6A4
SCHEMBL6233504 0.78 LOXL2 (0.56) CYP1A2CYP2A6CYP19A1CA2CA12
SCHEMBL1206769 0.78 CA2 (0.54) CYP1A2CYP2A6CA2CA12CA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952316-A FOR TREATING AUTOIMMUNE DISEASES, E.G., RHEUMATIOD ARTHRITIS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1999-09-14 US disclosed
US-5719176-A 2-amino-1,3-propanediol compound and immunosuppressant YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1998-02-17 US disclosed
US-5604229-A 2-amino-1,3-propanediol compound and immunosuppressant YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-02-18 US disclosed
EP-0627406-A1 2-AMINO-1,3-PROPANEDIOL COMPOUND AND IMMUNOSUPPRESSANT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-12-07 EP disclosed