SCHEMBL849960

SCHEMBL849960

N[C@H]([C]=O)Cc1ccc(O)c(O)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 8/20 0.59
KDM4E B2RXH2 7/20 0.59
HIF1A Q16665 6/20 0.59
HSD17B10 Q99714 6/20 0.59
RECQL P46063 5/20 0.59
TDP1 Q9NUW8 5/20 0.59
USP2 O75604 2/20 0.59
ADORA3 P0DMS8 2/20 0.59
HTR2A P28223 2/20 0.59
PTGS2 P35354 2/20 0.59
EGFR P00533 2/20 0.59
PTGS1 P23219 2/20 0.59
LCK P06239 1/20 0.59
FYN P06241 1/20 0.59
SLC7A5 Q01650 1/20 0.59
PLA2G1B P04054 1/20 0.55
ALOX12 P18054 5/20 0.53
MAPT P10636 5/20 0.53
MAPK1 P28482 4/20 0.53
ALDH1A1 P00352 4/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11136069 1.00 ALOX15 (0.59) ALOX15KDM4EHIF1AHSD17B10RECQL
SCHEMBL5311684 1.00 ALOX15 (0.59) ALOX15KDM4EHIF1AHSD17B10RECQL
SCHEMBL523986 0.84 THRB (0.44) ALOX15KDM4EHIF1AHSD17B10RECQL
SCHEMBL523987 0.84 THRB (0.44) ALOX15KDM4EHIF1AHSD17B10RECQL
SCHEMBL27734017 0.84 ALOX15 (0.42) ALOX15KDM4EHIF1AHSD17B10RECQL
SCHEMBL10412985 0.80 FOS (0.62) ALOX15TDP1PTGS1ALOX12MAPT
SCHEMBL10412984 0.80 FOS (0.62) ALOX15TDP1PTGS1ALOX12MAPT
SCHEMBL3985972 0.80 ALOX15 (0.43) ALOX15KDM4EHIF1AHSD17B10RECQL
SCHEMBL3985970 0.80 ALOX15 (0.43) ALOX15KDM4EHIF1AHSD17B10RECQL
SCHEMBL5144806 0.80 ALOX15 (0.40) ALOX15KDM4EHIF1AHSD17B10RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 593 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268678-B1 NOVEL 5-FLUOROURIDINE COMPOUNDS AND PROCESS FOR THEIR PREPARATION FUJI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1992-07-29 EP claimed
US-4892939-A ANTITUMOR, ANTIVIRAL AND IMMUNOSUPRESSIVE AGENTS FUJI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1990-01-09 US claimed
EP-0268678-A1 NOVEL 5-FLUOROURIDINE COMPOUNDS AND PROCESS FOR THEIR PREPARATION FUJI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1988-06-01 EP claimed
JP-61134397-A None JP disclosed
US-20240230669-A1 COMPOSITIONS AND METHODS FOR TREATING EYE INFECTIONS AND DISEASE UNIV VIRGINIA PATENT FOUNDATION (US) 2024-07-11 US disclosed
WO-2024121254-A1 LIGANDS SPECIFIC FOR ASCT1 METAFORA BIOSYSTEMS (FR) 2024-06-13 WO disclosed
US-20240148765-A1 COMPOSITIONS AND METHODS FOR TREATING AND/OR PREVENTING THERAPY-RELATED CARDIOMYOPATHY ASSOCIATED WITH NEUTROPHIL INFILTRATION UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2024-05-09 US disclosed
WO-2024078828-A1 CYTOTOXIC NECROTIZING FACTORS AS EXOGENOUS CARRIERS IN MAMMALIAN CELLS SE THERAPEUTICS (FR) 2024-04-18 WO disclosed
WO-2024052353-A1 PROXIMITY INDUCING SYSTEM AND USES THEREOF SORBONNE UNIVERSITE (FR) 2024-03-14 WO disclosed
WO-2024050285-A2 LEPTIN ANALOGS FOR TREATING OBESITY AND WEIGHT MANAGEMENT THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2024-03-07 WO disclosed
WO-2024030214-A2 BRINP2-DERIVED PEPTIDE COMPOSITIONS FOR TREATING OBESITY AND WEIGHT MANAGEMENT THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2024-02-08 WO disclosed
EP-0268678-B1 NOVEL 5-FLUOROURIDINE COMPOUNDS AND PROCESS FOR THEIR PREPARATION FUJI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1992-07-29 EP disclosed
US-4970297-A CONTAINING ISOXAZOLE RING SYNTEX (U.S.A.) INC. (US) 1990-11-13 US disclosed
US-4892939-A ANTITUMOR, ANTIVIRAL AND IMMUNOSUPRESSIVE AGENTS FUJI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1990-01-09 US disclosed
US-4892939-A ANTITUMOR, ANTIVIRAL AND IMMUNOSUPRESSIVE AGENTS FUJI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1990-01-09 US disclosed
EP-0268678-A1 NOVEL 5-FLUOROURIDINE COMPOUNDS AND PROCESS FOR THEIR PREPARATION FUJI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1988-06-01 EP disclosed
EP-0268678-A1 NOVEL 5-FLUOROURIDINE COMPOUNDS AND PROCESS FOR THEIR PREPARATION FUJI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1988-06-01 EP disclosed
WO-1987007276-A1 NOVEL 5-FLUOROURIDINE COMPOUNDS AND PROCESS FOR THEIR PREPARATION FUJI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1987-12-03 WO disclosed
JP-S61134397-A 5'-O-OLIGOPEPTIDYL-5-FLUOROURIDINE AND PRODUCTION THEREOF FUJI KAGAKU KOGYO KK 1986-06-21 JP disclosed
WO-1983002272-A1 SYNTHETIC PEPTIDES HAVING PITUITARY GROWTH HORMONE RELEASING ACTIVITY BECKMAN INSTRUMENTS INC (US) 1983-07-07 WO disclosed