SCHEMBL8500583

SCHEMBL8500583

NN=CNc1cccc(S(=O)(=O)Nc2cccc(-c3c(F)cc(F)cc3CCC(=O)O)c2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PFKFB3 Q16875 2/20 0.39
HSD17B1 P14061 3/20 0.38
HSD17B2 P37059 3/20 0.38
MAPT P10636 1/20 0.38
FFAR4 Q5NUL3 2/20 0.38
FFAR1 O14842 1/20 0.38
HTR6 P50406 2/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
MEN1 O00255 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
FABP1 P07148 1/20 0.37
AURKA O14965 1/20 0.37
AURKB Q96GD4 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4D Q08499 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8500575 0.88 MEN1 (0.42) PFKFB3HSD17B1HSD17B2MAPTFFAR4
SCHEMBL8499997 0.85 PFKFB3 (0.41) PFKFB3HSD17B1HSD17B2MAPTHTR6
SCHEMBL8501524 0.84 PFKFB3 (0.47) PFKFB3HSD17B1HSD17B2MAPTPTGDR2
SCHEMBL8501758 0.81 HTR6 (0.43) PFKFB3HSD17B1HSD17B2MAPTFFAR1
SCHEMBL8500619 0.81 ALDH1A1 (0.49) MAPTMEN1HPGDKMT2ASMN1; SMN2
SCHEMBL7376815 0.77 ALDH1A1 (0.55) MAPTFFAR4FFAR1HTR6MEN1
SCHEMBL8499992 0.74 MEN1 (0.42) PFKFB3HSD17B1HSD17B2MAPTMEN1
SCHEMBL7861775 0.74 EEF2K (0.43) PFKFB3MAPTHTR6MEN1HPGD
SCHEMBL8536202 0.73 FFAR1 (0.35) MAPTFFAR4FFAR1PTGDR2HPGD
SCHEMBL8496957 0.73 MEN1 (0.43) PFKFB3HSD17B1HSD17B2MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP disclosed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO disclosed