SCHEMBL8501758

SCHEMBL8501758

NN=CNc1cccc(S(=O)(=O)Nc2cccc(-c3cc(CCC(=O)O)ccc3F)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.43
HSD17B1 P14061 3/20 0.40
HSD17B2 P37059 3/20 0.40
PFKFB3 Q16875 2/20 0.40
PARP1 P09874 1/20 0.40
ALDH1A1 P00352 1/20 0.40
FFAR1 O14842 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
NPY1R P25929 1/20 0.39
NPY2R P49146 1/20 0.39
FABP4 P15090 1/20 0.39
PLA2G10 O15496 1/20 0.39
PLA2G2A P14555 1/20 0.39
SLCO1B1 Q9Y6L6 1/20 0.39
ERAP1 Q9NZ08 1/20 0.39
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8501754 0.88 MEN1 (0.44) HTR6HSD17B1HSD17B2PFKFB3PARP1
SCHEMBL7376815 0.85 ALDH1A1 (0.55) HTR6ALDH1A1FFAR1MEN1KMT2A
SCHEMBL8501524 0.84 PFKFB3 (0.47) HSD17B1HSD17B2PFKFB3MEN1KMT2A
SCHEMBL8499997 0.83 PFKFB3 (0.41) HTR6HSD17B1HSD17B2PFKFB3MEN1
SCHEMBL8500583 0.81 PFKFB3 (0.39) HTR6HSD17B1HSD17B2PFKFB3FFAR1
SCHEMBL8371225 0.79 ITGB3 (0.53) HTR6PFKFB3MEN1KMT2AMAPT
SCHEMBL8500892 0.74 PTGDR2 (0.35) HTR6PFKFB3ALDH1A1MEN1KMT2A
SCHEMBL8371139 0.72 ITGB3 (0.57) HTR6ALDH1A1MEN1KMT2APOLB
SCHEMBL14532378 0.72 ITGB3 (0.57) HTR6ALDH1A1MEN1KMT2APOLB
SCHEMBL7864756 0.72 CA1 (0.38) HTR6HSD17B1HSD17B2PFKFB3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed