SCHEMBL8501462

SCHEMBL8501462

CCC(=O)Oc1ccc(Oc2c(-c3ccc(O)cc3)ccc3cc(OC)ccc23)cc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 16/20 0.47
ESR2 Q92731 14/20 0.47
XDH P47989 1/20 0.41
BACE1 P56817 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TP53 P04637 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8497579 0.94 SMN1; SMN2 (0.42) ESR1ESR2BACE1KDM4ETP53
SCHEMBL8497550 0.94 ESR1 (0.49) ESR1ESR2BACE1KDM4EMEN1
SCHEMBL8499778 0.92 ESR1 (0.54) ESR1ESR2MAPTKMT2A
SCHEMBL8501430 0.90 ESR1 (0.46) ESR1ESR2KDM4EALDH1A1MAPT
SCHEMBL8501243 0.90 KDM4E (0.39) ESR1ESR2KDM4EMEN1ALDH1A1
SCHEMBL8497702 0.89 ESR1 (0.49) ESR1ESR2MEN1CYP3A4CYP2D6
SCHEMBL8500568 0.88 ESR1 (0.48) ESR1ESR2MEN1KMT2A
SCHEMBL8502205 0.87 MTNR1A (0.43) ESR1ESR2CYP3A4CYP2D6CYP2C9
SCHEMBL8497879 0.87 KMT2A (0.42) ESR1ESR2BACE1KDM4EALDH1A1
SCHEMBL8497867 0.86 ESR1 (0.57) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed