SCHEMBL8501774

SCHEMBL8501774

CN(C=O)c1ccc(Br)s1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
DAO P14920 1/20 0.33
GSK3B P49841 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9943768 0.69 DAO (0.45) KDM4EALDH1A1KMT2ACES2CES1
SCHEMBL2742897 0.67 KDM4E (0.45) KDM4EALDH1A1KMT2A
SCHEMBL722021 0.66 CES2 (0.32) CES2CES1
SCHEMBL724067 0.65 L3MBTL1 (0.30)
SCHEMBL722509 0.65 ATM (0.33)
SCHEMBL209431 0.64
SCHEMBL2090725 0.62 MAPT (0.40) KDM4EALDH1A1KMT2ACES2CES1
SCHEMBL16539971 0.62 ALDH1A1 (0.42) ALDH1A1KMT2ADAO
SCHEMBL147222 0.61
SCHEMBL50975 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939398-A ANTIATHEROSCLEROSIS AGENTS PFIZER INC. (US) 1999-08-17 US disclosed