SCHEMBL8506958

SCHEMBL8506958

O=C1C(Br)CCN1CC1CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 2/20 0.45
ADRA2C P18825 1/20 0.45
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM1 P11229 1/20 0.36
ACHE P22303 1/20 0.36
OPRM1 P35372 2/20 0.36
OPRL1 P41146 2/20 0.36
HSD11B1 P28845 1/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
MMP1 P03956 4/20 0.35
MMP9 P14780 3/20 0.35
MMP7 P09237 2/20 0.35
MMP3 P08254 1/20 0.35
TRPC5 Q9UL62 1/20 0.35
DRD2 P14416 2/20 0.35
SIGMAR1 Q99720 2/20 0.35
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7510369 0.90 FPR2 (0.35) CHRM5ADRA2C
SCHEMBL7619075 0.90 FPR2 (0.35) CHRM5ADRA2C
SCHEMBL7619079 0.90 FPR2 (0.35) CHRM5ADRA2C
SCHEMBL6964128 0.78 FPR2 (0.38) SMN1; SMN2
SCHEMBL4227086 0.78 CHRM5 (0.45) CHRM5ADRA2CCHRM2CHRM4CHRM1
SCHEMBL892512 0.74 CHRM5 (0.41) CHRM5ADRA2CSMN1; SMN2
SCHEMBL8560638 0.73 MAPT (0.51)
SCHEMBL8900108 0.73 MAPT (0.51)
SCHEMBL8560636 0.73 MAPT (0.51)
SCHEMBL2083375 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5925632-A BACTERICIDES HOFFMANN-LA ROCHE INC. (US) 1999-07-20 US disclosed
CN-1176641-A Derivatives of 3-pyrrolidylidene -2 -one -cephalosporines HOFFMANN LA ROCHE (CH) 1998-03-18 CN disclosed
EP-0812323-A1 DERIVATIVES OF 3-PYRROLIDYLIDENE-2-ONE-CEPHALOSPORINES F. HOFFMANN-LA ROCHE AG (CH) 1997-12-17 EP disclosed
WO-1996026943-A1 DERIVATIVES OF 3-PYRROLIDYLIDENE-2-ONE-CEPHALOSPORINES F.HOFFMANN-LA ROCHE AG (CH) 1996-09-06 WO disclosed