SCHEMBL8510671

SCHEMBL8510671

CC(C)Oc1ccc(-c2ccnc(N3CCC(O)CC3)n2)cc1C(C)(C)C

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DKK1 O94907 3/20 0.44
KMO O15229 1/20 0.43
MTOR P42345 1/20 0.40
LRRK2 Q5S007 3/20 0.39
EGFR P00533 3/20 0.38
PIK3CA P42336 1/20 0.38
SORD Q00796 1/20 0.38
ITGB2 P05107 2/20 0.38
ICAM1 P05362 2/20 0.38
ITGAL P20701 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8512439 0.91 DKK1 (0.56) DKK1KMOMTORPIK3CASORD
Hydrochloric Acid SCHEMBL8513412 0.90 DKK1 (0.55) DKK1KMOMTORPIK3CASORD
SCHEMBL8514134 0.89 DKK1 (0.42) DKK1KMOMTOREGFRPIK3CA
SCHEMBL8510840 0.89 KMO (0.43) DKK1KMOMTORLRRK2PIK3CA
SCHEMBL8511678 0.88 DKK1 (0.58) DKK1KMOMTORPIK3CASORD
SCHEMBL8514794 0.88 DKK1 (0.41) DKK1KMOMTORLRRK2PIK3CA
Ammonia Solution, Strong SCHEMBL8587136 0.87 DYRK1A (0.43) DKK1KMOSORD
SCHEMBL8515838 0.87 DKK1 (0.49) DKK1KMOLRRK2
SCHEMBL8511790 0.87 ROCK2 (0.41) DKK1KMOLRRK2EGFRPIK3CA
SCHEMBL9612712 0.86 DKK1 (0.40) DKK1KMOMTORLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed