SCHEMBL8510708

SCHEMBL8510708

CC1(C)CCC(C)(C)c2cc(-c3nccc(OC4CCN(C(=O)O)CC4)n3)ccc21

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RARB P10826 14/20 0.42
RARA P10276 13/20 0.42
RARG P13631 14/20 0.42
RXRA P19793 4/20 0.39
ABCB1 P08183 1/20 0.38
ABCC1 P33527 1/20 0.38
FFAR4 Q5NUL3 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8511463 0.81 SYK (0.43) RARBRARARARG
Trifluoroacetic Acid SCHEMBL8511882 0.81 RARB (0.39) RARBRARARARGRXRAABCB1
SCHEMBL8515150 0.75 EPHX2 (0.41)
SCHEMBL8514108 0.72 CHEK2 (0.44)
SCHEMBL8515197 0.71 RARB (0.42) RARBRARARARGRXRAABCB1
SCHEMBL8513291 0.70 GPR119 (0.52)
SCHEMBL16612996 0.69 RARA (0.47) RARBRARARARGRXRAABCB1
SCHEMBL5267332 0.69 MALT1 (0.45)
SCHEMBL14121158 0.68 SPR (0.40)
SCHEMBL30757104 0.68 SPR (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed