SCHEMBL8510980

SCHEMBL8510980

CC(C)Oc1ccc(Br)cc1C(C)(C)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.42
LMNA P02545 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
ALDH1A1 P00352 2/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42
ALOX12 P18054 1/20 0.42
HTT P42858 1/20 0.42
AR P10275 1/20 0.36
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36
AAK1 Q2M2I8 4/20 0.35
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
MAPK1 P28482 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8510244 0.86 LMNA (0.39) PTGDR2LMNASMN1; SMN2ALDH1A1POLB
SCHEMBL8515160 0.86 PTGDR2 (0.51) PTGDR2LMNASMN1; SMN2ALDH1A1POLB
SCHEMBL30597890 0.81 RXRA (0.49) PTGDR2LMNASMN1; SMN2ALDH1A1POLB
SCHEMBL1293281 0.81 RXRA (0.49) PTGDR2LMNASMN1; SMN2ALDH1A1POLB
SCHEMBL4820133 0.80 PTGDR2 (0.45) PTGDR2LMNASMN1; SMN2ALDH1A1MAPT
SCHEMBL17703261 0.76 PTGDR2 (0.42) PTGDR2LMNASMN1; SMN2ALDH1A1MAPT
SCHEMBL2284093 0.76 ALDH1A1 (0.43) LMNASMN1; SMN2ALDH1A1POLBMAPT
SCHEMBL1330449 0.74 SLC6A4 (0.49) LMNASMN1; SMN2ALDH1A1POLBMAPT
SCHEMBL9259271 0.74 MAPK1 (0.58) LMNASMN1; SMN2ALDH1A1POLBMAPT
SCHEMBL7847441 0.73 PTGDR2 (0.40) PTGDR2ALDH1A1HTTRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed