SCHEMBL8513449

SCHEMBL8513449

CC(C)Oc1ccc(-c2ncnc(N3CCNCC3)n2)cc1C(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 3/20 0.42
HRH4 Q9H3N8 1/20 0.40
ALDH1A1 P00352 4/20 0.36
CYP1A2 P05177 3/20 0.36
PIK3CA P42336 2/20 0.36
USP2 O75604 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C19 P33261 2/20 0.36
CLK4 Q9HAZ1 1/20 0.36
LRRK2 Q5S007 1/20 0.36
KHK P50053 1/20 0.35
TGFBR1 P36897 1/20 0.35
ACVR1 Q04771 1/20 0.35
TLR9 Q9NR96 1/20 0.35
TLR8 Q9NR97 1/20 0.35
TLR7 Q9NYK1 1/20 0.35
ADRB1 P08588 1/20 0.35
JAK2 O60674 1/20 0.35
TBK1 Q9UHD2 1/20 0.35
EGFR P00533 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8510076 0.99 S1PR1 (0.41) S1PR1HRH4ALDH1A1CYP1A2PIK3CA
SCHEMBL8514773 0.83 ADRB1 (0.43) S1PR1ALDH1A1PIK3CACLK4ADRB1
Hydrochloric Acid SCHEMBL8514967 0.82 ADRB1 (0.42) S1PR1ALDH1A1CLK4ADRB1TBK1
SCHEMBL8512449 0.80 PIK3CA (0.46) PIK3CATLR9TLR7
SCHEMBL8511499 0.75 S1PR1 (0.43) S1PR1ALDH1A1PIM1PIM3PIM2
Hydrochloric Acid SCHEMBL8512803 0.74 S1PR1 (0.42) S1PR1ALDH1A1PIM1PIM3PIM2
SCHEMBL19124978 0.71 CETP (0.56) HRH4ALDH1A1CYP1A2USP2CYP3A4
SCHEMBL2035508 0.70 HRH4 (0.43) HRH4ALDH1A1CYP1A2PIK3CACYP3A4
SCHEMBL8511517 0.70 CYP1A2 (0.40) ALDH1A1CYP1A2PIK3CAUSP2CYP3A4
SCHEMBL8511790 0.68 ROCK2 (0.41) S1PR1ALDH1A1PIK3CACLK4LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed