SCHEMBL8511699

SCHEMBL8511699

CC1(C)CCC(C)(C)c2cc(-c3ccnc(OC4CCNCC4)n3)ccc21.Cc1nc(-c2ccc3c(c2)C(C)(C)CCC3(C)C)cc(N2CCNCC2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.41
PRKD1 Q15139 14/20 0.38
PRKD2 Q9BZL6 13/20 0.38
KMT2A Q03164 1/20 0.34
KARS1 Q15046 2/20 0.34
PRKD3 O94806 2/20 0.34
EGFR P00533 1/20 0.34
PRKCG P05129 1/20 0.34
PRKCB P05771 1/20 0.34
LCK P06239 1/20 0.34
PRKCA P17252 1/20 0.34
PRKCH P24723 1/20 0.34
PRKCI P41743 1/20 0.34
ZAP70 P43403 1/20 0.34
PRKCE Q02156 1/20 0.34
PRKCQ Q04759 1/20 0.34
PRKCZ Q05513 1/20 0.34
PRKCD Q05655 1/20 0.34
ADRB1 P08588 1/20 0.34
BRD4 O60885 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8510098 0.93 IRAK4 (0.36) IRAK4PRKD1PRKD2KARS1PRKD3
SCHEMBL8511070 0.86 IRAK4 (0.48) IRAK4PRKD3PRKCBPRKCABRD4
SCHEMBL9612709 0.83 KMT2A (0.47) PRKD1PRKD2KMT2AKARS1PRKD3
Trifluoroacetic Acid SCHEMBL8514001 0.78 RARA (0.42) IRAK4MAPK14
Trifluoroacetic Acid SCHEMBL8537644 0.75 HRH4 (0.43) PRKD1PRKD2KMT2APRKD3
SCHEMBL8512407 0.73 ADRB1 (0.44) KMT2AADRB1
Hydrochloric Acid SCHEMBL8512430 0.72 ADRB1 (0.43) KMT2AADRB1
SCHEMBL2016664 0.71 DYRK1A (0.54) PRKD1PRKD2KARS1PRKD3ADRB1
SCHEMBL8515571 0.70 CYP1A2 (0.47) PRKD1PRKD2KMT2APRKD3ADRB1
SCHEMBL8514909 0.70 CYP1A2 (0.52) DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed