SCHEMBL9612709

SCHEMBL9612709

Cc1nc(-c2ccc3c(c2)C(C)(C)CCC3(C)C)cc(N2CCNCC2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.47
HRH4 Q9H3N8 2/20 0.44
HRH3 Q9Y5N1 1/20 0.44
ADRB1 P08588 1/20 0.40
NCF1 P14598 1/20 0.40
RARA P10276 3/20 0.39
RARB P10826 3/20 0.39
CASP1 P29466 1/20 0.38
CASP4 P49662 1/20 0.38
CASP5 P51878 1/20 0.38
CYP1A2 P05177 1/20 0.38
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
HTR2C P28335 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
UBE2N P61088 1/20 0.37
PRKD1 Q15139 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8537644 0.90 HRH4 (0.43) KMT2AHRH4HRH3RARARARB
SCHEMBL8511699 0.83 IRAK4 (0.41) KMT2AADRB1PRKD1PRKD2PRKD3
SCHEMBL8514909 0.81 CYP1A2 (0.52) HRH4RARARARBCYP1A2KDM4E
SCHEMBL2014630 0.81 RARA (0.51) RARARARBALDH1A1KARS1
SCHEMBL8514715 0.81 RARA (0.46) KMT2ARARARARBRARG
Hydrochloric Acid SCHEMBL8512697 0.81 CYP1A2 (0.51) HRH4RARARARBCYP1A2KDM4E
SCHEMBL8514096 0.81 ROCK2 (0.55) KMT2ARARARARBCYP1A2ROCK2
Hydrochloric Acid SCHEMBL8515528 0.80 ROCK2 (0.54) KMT2AADRB1CYP1A2ROCK2ROCK1
SCHEMBL2013665 0.78 IRAK4 (0.49) RARARARBROCK2ROCK1ALDH1A1
SCHEMBL8510098 0.78 IRAK4 (0.36) ADRB1PRKD1PRKD2PRKD3KARS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed