SCHEMBL8512804

SCHEMBL8512804

CC1(C)CCC(C)(C)c2cc(-c3ccnc(-c4cccnc4)n3)ccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 3/20 0.49
RARB P10826 3/20 0.49
CYP1A2 P05177 8/20 0.44
CYP3A4 P08684 7/20 0.44
CYP2D6 P10635 6/20 0.44
CLK4 Q9HAZ1 4/20 0.44
ALDH1A1 P00352 3/20 0.44
HSD17B10 Q99714 3/20 0.44
TSHR P16473 2/20 0.44
CYP2A6 P11509 2/20 0.44
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
PTK2 Q05397 1/20 0.43
RARG P13631 2/20 0.43
MAPKAPK2 P49137 4/20 0.43
CYP2C19 P33261 4/20 0.42
ALOX15 P16050 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ammonia Solution, Strong SCHEMBL8514741 0.86 CYP1A2 (0.53) RARARARBCYP1A2CYP3A4CYP2D6
SCHEMBL8514253 0.84 NPC1 (0.55) RARARARBCYP1A2CYP3A4CYP2D6
SCHEMBL8511483 0.77 RARB (0.46) RARARARBCYP3A4ALDH1A1RARG
SCHEMBL8510213 0.76 RARA (0.50) RARARARBALDH1A1RARGKDM4E
SCHEMBL31060783 0.76 RARB (0.51) RARARARBRARGMEN1NPC1
SCHEMBL8515254 0.76 RARB (0.51) RARARARBRARGMEN1NPC1
SCHEMBL8511696 0.75 RARB (0.44) RARARARBRARGSMN1; SMN2KDM4E
SCHEMBL9612772 0.75 RARB (0.47) RARARARBCYP3A4RARGMEN1
Hydrochloric Acid SCHEMBL8515237 0.74 RARB (0.44) RARARARBRARGSMN1; SMN2KDM4E
SCHEMBL18905348 0.74 CYP2A6 (0.62) CYP1A2CYP3A4CYP2D6CLK4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed