SCHEMBL8510213

SCHEMBL8510213

CC1(C)CCC(C)(C)c2cc(-c3ccnc(Cl)n3)ccc21

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RARA P10276 12/20 0.50
RARB P10826 11/20 0.50
RARG P13631 11/20 0.43
RXRA P19793 3/20 0.42
KMO O15229 3/20 0.40
ABCB1 P08183 1/20 0.39
ABCC1 P33527 1/20 0.39
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
CYP26A1 O43174 1/20 0.35
CYP26B1 Q9NR63 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8514253 0.81 NPC1 (0.55) RARARARBRARGRXRAABCB1
SCHEMBL2015591 0.79 RARA (0.44) RARARARBRARGRXRAABCB1
SCHEMBL18961191 0.79 RARA (0.47) RARARARBRARGRXRAABCB1
SCHEMBL8511483 0.76 RARB (0.46) RARARARBRARGRXRAKMO
SCHEMBL8512804 0.76 RARA (0.49) RARARARBRARGKDM4EALDH1A1
SCHEMBL16998453 0.76 CCR1 (0.50) RARARARBRARGRXRAABCB1
SCHEMBL29666144 0.76 KMO (0.35) KMOKDM4EALDH1A1POLB
SCHEMBL31060783 0.76 RARB (0.51) RARARARBRARGRXRAABCB1
SCHEMBL8515254 0.76 RARB (0.51) RARARARBRARGRXRAABCB1
SCHEMBL8512407 0.74 ADRB1 (0.44) RARARARBKDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed