SCHEMBL8513596

SCHEMBL8513596

O=C1c2ccccc2OC2C=CN=CC12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.36
KDR P35968 1/20 0.36
MEN1 O00255 2/20 0.36
POLB P06746 2/20 0.36
KMT2A Q03164 2/20 0.36
STK17B O94768 1/20 0.35
CYP19A1 P11511 6/20 0.34
MAOB P27338 2/20 0.34
ADORA3 P0DMS8 2/20 0.34
AR P10275 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HSD17B10 Q99714 1/20 0.34
PKM P14618 1/20 0.33
TSHR P16473 1/20 0.33
PARP1 P09874 1/20 0.32
NFKB1 P19838 1/20 0.32
STAT3 P40763 1/20 0.32
STAT1 P42224 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30891245 0.77 RET (0.40) RETKDRMEN1POLBKMT2A
SCHEMBL11380880 0.77 RET (0.40) RETKDRMEN1POLBKMT2A
SCHEMBL22146506 0.68 MAOB (0.38) RETKDRMEN1POLBKMT2A
SCHEMBL5548145 0.64 RET (0.46) RETKDRMEN1POLBKMT2A
SCHEMBL11741033 0.64 S100A4 (0.56) RETKDRMEN1POLBKMT2A
SCHEMBL69430 0.63 PARP1 (0.48) RETKDRMEN1POLBKMT2A
SCHEMBL69727 0.63 RET (0.53) RETKDRMEN1POLBKMT2A
SCHEMBL4775874 0.63 RET (0.45) RETKDRMEN1POLBKMT2A
SCHEMBL1429502 0.63 STK17B (0.46) RETKDRMEN1POLBKMT2A
SCHEMBL29441433 0.61 MEN1 (0.52) RETKDRMEN1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012071458-A1 HETEROCYCLIC INHIBITORS OF BETA - SECRETASE FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES ARRAY BIOPHARMA INC. (US) 2012-05-31 WO disclosed