SCHEMBL8514383

SCHEMBL8514383

Cc1[nH]nc(O)c1CC(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
LMNA P02545 1/20 0.42
GABRR1 P24046 1/20 0.39
KDM4E B2RXH2 4/20 0.39
MAPT P10636 4/20 0.39
GAA P10253 3/20 0.39
ALDH1A1 P00352 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
HCAR2 Q8TDS4 3/20 0.38
DAO P14920 1/20 0.38
CSNK2A2 P19784 1/20 0.37
CSNK2B P67870 1/20 0.37
CSNK2A1 P68400 1/20 0.37
CSNK2A3 Q8NEV1 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2830618 0.82 MEN1 (0.51) MEN1KMT2ALMNAKDM4EPDE4D
Hydrochloric Acid SCHEMBL1375056 0.80 MEN1 (0.50) MEN1KMT2ALMNAKDM4EPDE4D
SCHEMBL14556062 0.76 KDM4E (0.40) MEN1KMT2ALMNAGABRR1KDM4E
SCHEMBL4362757 0.72 MEN1 (0.39) MEN1KMT2ALMNAGABRR1KDM4E
SCHEMBL8515102 0.72 RAB9A (0.49) LMNAKDM4EMAPTGAAALDH1A1
SCHEMBL14487981 0.69 GABRR1 (0.48) MEN1KMT2ALMNAGABRR1KDM4E
SCHEMBL8801602 0.68 CYP1A2 (0.40) MEN1KMT2ALMNAGABRR1KDM4E
SCHEMBL4350884 0.68 LMNA (0.39) MEN1KMT2ALMNAGABRR1KDM4E
SCHEMBL4362752 0.67 MEN1 (0.38) MEN1KMT2ALMNAGABRR1KDM4E
SCHEMBL31358629 0.67 HCAR2 (0.40) MEN1KMT2ALMNAKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069175-A1 NEW PYRAZOLE DERIVATIVES HAVING CRTH2 ANTAGONISTIC BEHAVIOUR ALMIRALL, S.A. (ES) 2012-05-31 WO disclosed
EP-2457900-A1 New pyrazole derivatives having CRTh2 antagonistic behaviour Almirall, S.A. (ES) 2012-05-30 EP disclosed