SCHEMBL8514744

SCHEMBL8514744

CC(C)Oc1ccc(-c2cccc(N3CCNCC3)n2)cc1C(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.41
KARS1 Q15046 4/20 0.40
PRKCA P17252 1/20 0.40
PRKCQ Q04759 1/20 0.40
PRKCD Q05655 1/20 0.40
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
PIM1 P11309 10/20 0.39
PRKD1 Q15139 1/20 0.39
PRKD2 Q9BZL6 1/20 0.39
PIM3 Q86V86 3/20 0.38
PIM2 Q9P1W9 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8512940 0.99 S1PR1 (0.41) S1PR1KARS1PRKCAPRKCQPRKCD
SCHEMBL8510804 0.87 PIM1 (0.42) KARS1PRKCAPRKCQPRKCDPIM1
Hydrochloric Acid SCHEMBL8514424 0.86 PIM1 (0.41) KARS1PRKCAPRKCQPRKCDPIM1
SCHEMBL8511499 0.85 S1PR1 (0.43) S1PR1KARS1PRKCAPRKCQPRKCD
Hydrochloric Acid SCHEMBL8512803 0.84 S1PR1 (0.42) S1PR1KARS1PRKCAPRKCQPRKCD
SCHEMBL8514718 0.83 KARS1 (0.46) KARS1PRKCAPRKCQPRKCDPIM1
SCHEMBL8514667 0.83 KARS1 (0.41) S1PR1KARS1PRKCAPRKCQPRKCD
Hydrochloric Acid SCHEMBL8511433 0.82 KARS1 (0.45) KARS1PRKCAPRKCQPRKCDPIM1
SCHEMBL8511790 0.82 ROCK2 (0.41) S1PR1PRKCAPRKCQPRKCDALDH1A1
Hydrochloric Acid SCHEMBL8513958 0.82 KARS1 (0.41) S1PR1KARS1PRKCAPRKCQPRKCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed