SCHEMBL8516080

SCHEMBL8516080

CCN(CC)C(=O)C(OC(=O)C(F)(F)F)n1cc(-c2nc3cc(Cl)c(Cl)cc3n(CCCN)c2=O)c2ccccc21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 10/20 0.35
CYP1A2 P05177 10/20 0.35
CYP3A4 P08684 8/20 0.35
CYP2C9 P11712 6/20 0.35
CYP2C19 P33261 4/20 0.35
ALDH1A1 P00352 2/20 0.35
CLK4 Q9HAZ1 1/20 0.35
CASP1 P29466 7/20 0.33
CASP7 P55210 7/20 0.33
MEN1 O00255 5/20 0.33
KMT2A Q03164 5/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 2/20 0.32
HBB P68871 3/20 0.32
TSHR P16473 3/20 0.31
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
TYK2 P29597 1/20 0.31
JAK3 P52333 1/20 0.31
LMNA P02545 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517087 0.98 USP2 (0.34) USP2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8516522 0.93 USP2 (0.33) USP2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8516687 0.92 USP2 (0.33) USP2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8365258 0.91 ALDH1A1 (0.37) USP2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8516861 0.89 ALDH1A1 (0.36) USP2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8367898 0.88 CTSB (0.31) USP2CYP1A2CYP3A4CASP1CASP7
SCHEMBL8516657 0.87 PDE4B (0.32)
SCHEMBL8365344 0.84 ATM (0.39) USP2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8365273 0.83 BRD4 (0.37) ALDH1A1LMNAHIF1A
SCHEMBL8365239 0.82 MAPT (0.38) USP2CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999046260-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 1999-09-16 WO claimed