SCHEMBL8516372

SCHEMBL8516372

CCCCCCCCCCc1nnc(Br)c(-c2ccccc2)c1-c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.52
GCGR P47871 2/20 0.45
GPR84 Q9NQS5 1/20 0.43
HSD11B1 P28845 2/20 0.42
KCNH2 Q12809 2/20 0.38
TSHR P16473 1/20 0.37
CYP19A1 P11511 6/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
SOAT1 P35610 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15068306 0.75 GCGR (0.53) DHFRGCGRGPR84HSD11B1SOAT1
SCHEMBL15068263 0.75 GCGR (0.53) DHFRGCGRGPR84HSD11B1SOAT1
SCHEMBL15068264 0.70 GPR84 (0.63) DHFRGCGRGPR84HSD11B1KCNH2
SCHEMBL15068307 0.70 GPR84 (0.63) DHFRGCGRGPR84HSD11B1KCNH2
SCHEMBL1754697 0.70 DHFR (0.46) DHFRGCGRGPR84HSD11B1TSHR
SCHEMBL6512533 0.70 GCGR (0.54) DHFRGCGRGPR84HSD11B1KCNH2
SCHEMBL28111153 0.70 GCGR (0.58) DHFRGCGRGPR84HSD11B1KCNH2
SCHEMBL9128219 0.69 LIPG (0.47) DHFRGCGR
SCHEMBL4838823 0.69 DHFR (1.00) DHFR
SCHEMBL16678699 0.68 HSD11B1 (0.63) HSD11B1KCNH2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628530-B1 ACETYLENE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL CO (JP) 1999-03-24 EP disclosed
US-5534188-A Acetylene derivatives, process for producing the same, liquid crystal composition containing the same as an active ingredient, and liquid crystal element using said liquid crystal composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-07-09 US disclosed
EP-0628530-A1 ACETYLENE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-12-14 EP disclosed