SCHEMBL8516502

SCHEMBL8516502

C=CCc1ccccc1-c1cnc(C#CC(C)O)nc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 6/20 0.39
ADRB1 P08588 4/20 0.39
LMNA P02545 2/20 0.39
ADRB3 P13945 2/20 0.39
ADRA2C P18825 2/20 0.39
HTR1A P08908 1/20 0.39
SLC6A2 P23975 1/20 0.39
BDKRB2 P30411 1/20 0.39
SLC6A4 P31645 1/20 0.39
ADRA1A P35348 1/20 0.39
HTR2B P41595 1/20 0.39
KCNH2 Q12809 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
KDM4E B2RXH2 1/20 0.39
PMP22 Q01453 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517500 0.80 ADRB2 (0.39) ADRB2ADRB1LMNAADRB3ADRA2C
SCHEMBL9287495 0.70 GABRA1 (0.42) KDM4EGABRA1GABRB2KMT2AAKR1B1
SCHEMBL8517770 0.70 ADRB2 (0.32) ADRB2ADRB1LMNAADRB3ADRA2C
SCHEMBL8517938 0.70 ADRB2 (0.34) ADRB2ADRB1LMNAADRB3ADRA2C
SCHEMBL7865025 0.69 GABRA1 (0.41) ADRB2ADRB1LMNAADRB3ADRA2C
SCHEMBL9287653 0.67 HIF1A (0.41) KDM4EALDH1A1GABRA1GABRB2AKR1B1
SCHEMBL8517808 0.67 ALDH1A1 (0.36) LMNATSHRKDM4EALDH1A1GABRA1
SCHEMBL170787 0.66 DPP4 (0.54) ADRB2ADRB1KCNH2KDM4EALDH1A1
SCHEMBL6537109 0.66 GABRA1 (0.59) ADRB2ADRB1LMNACYP1A2CYP2D6
SCHEMBL27744825 0.66 GABRA1 (0.50) ADRB2ADRB1ADRA2CALDH1A1GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628530-B1 ACETYLENE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL CO (JP) 1999-03-24 EP disclosed
US-5534188-A Acetylene derivatives, process for producing the same, liquid crystal composition containing the same as an active ingredient, and liquid crystal element using said liquid crystal composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-07-09 US disclosed
EP-0628530-A1 ACETYLENE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-12-14 EP disclosed