SCHEMBL8517666

SCHEMBL8517666

C=CCOc1ccc2nc(C#CC(C)O)ncc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.40
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MAPT P10636 2/20 0.37
ALDH1A1 P00352 2/20 0.37
GAA P10253 2/20 0.37
CA12 O43570 4/20 0.36
CA1 P00915 4/20 0.36
CA9 Q16790 4/20 0.36
CASR P41180 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SRC P12931 2/20 0.35
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35
ADRB3 P13945 1/20 0.35
ABL1 P00519 1/20 0.35
HPGD P15428 3/20 0.34
FGFR1 P11362 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517808 0.81 ALDH1A1 (0.36) LMNASMN1; SMN2NPSR1MAPTALDH1A1
SCHEMBL8517796 0.79 CYP2D6 (0.43) CYP2D6LMNASMN1; SMN2NPSR1MAPT
SCHEMBL8517137 0.78 CYP2D6 (0.48) CYP2D6LMNASMN1; SMN2MAPTALDH1A1
SCHEMBL8517269 0.77 CYP2D6 (0.35) CYP2D6LMNASMN1; SMN2NPSR1ADRB2
SCHEMBL8517692 0.73 ADRB2 (0.39) CYP2D6ALDH1A1GAAMEN1KMT2A
SCHEMBL8051440 0.71 PDE3B (0.43) CYP2D6LMNASMN1; SMN2NPSR1MAPT
SCHEMBL8051435 0.71 PDE3B (0.43) CYP2D6LMNASMN1; SMN2NPSR1MAPT
SCHEMBL8517707 0.71 CYP2D6 (0.51) CYP2D6LMNASMN1; SMN2MAPTALDH1A1
SCHEMBL8517181 0.70 CYP2D6 (0.45) CYP2D6MAPTALDH1A1GAACA12
SCHEMBL8517467 0.70 LMNA (0.40) CYP2D6LMNASMN1; SMN2NPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628530-B1 ACETYLENE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL CO (JP) 1999-03-24 EP disclosed
US-5534188-A Acetylene derivatives, process for producing the same, liquid crystal composition containing the same as an active ingredient, and liquid crystal element using said liquid crystal composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-07-09 US disclosed
EP-0628530-A1 ACETYLENE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-12-14 EP disclosed