SCHEMBL851771

SCHEMBL851771

Oc1ccc(-c2ccccc2)nc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.57
CYP11B1 P15538 5/20 0.51
CYP11B2 P19099 5/20 0.51
HSD17B1 P14061 2/20 0.50
HSD17B2 P37059 2/20 0.50
BAZ2B Q9UIF8 1/20 0.49
MEN1 O00255 1/20 0.48
NTSR1 P30989 1/20 0.48
KMT2A Q03164 1/20 0.48
MMP3 P08254 1/20 0.48
BCL2L1 Q07817 1/20 0.48
MKNK1 Q9BUB5 1/20 0.47
MKNK2 Q9HBH9 1/20 0.47
CYP2C8 P10632 1/20 0.47
CYP2C9 P11712 1/20 0.47
HCAR2 Q8TDS4 1/20 0.47
HPGDS O60760 2/20 0.46
IDO1 P14902 1/20 0.46
TDO2 P48775 1/20 0.46
BCHE P06276 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29392609 1.00 LDHA (0.57) LDHACYP11B1CYP11B2HSD17B1HSD17B2
SCHEMBL18573277 0.96 MMP3 (0.56) LDHACYP11B1CYP11B2HSD17B1HSD17B2
SCHEMBL21477415 0.81 ABL1 (0.53) LDHACYP11B1CYP11B2HSD17B1HSD17B2
SCHEMBL28326772 0.80 CYP11B1 (0.44) CYP11B1CYP11B2HSD17B1HSD17B2IDO1
SCHEMBL1070654 0.80 CCR1 (0.46) HSD17B1HSD17B2MEN1KMT2ABCHE
SCHEMBL30958843 0.80 CCR1 (0.46) HSD17B1HSD17B2MEN1KMT2ABCHE
Phenol SCHEMBL27328542 0.79 HSD17B1 (0.65) LDHACYP11B1CYP11B2HSD17B1HSD17B2
SCHEMBL2435669 0.78 NPC1 (0.58) CYP11B1CYP11B2HSD17B1HSD17B2MEN1
SCHEMBL8592351 0.78 MEN1 (0.53) HSD17B1HSD17B2MEN1KMT2ACYP2C8
SCHEMBL2435624 0.78 MAPT (0.53) HSD17B1HSD17B2MEN1KMT2ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 97 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248488-A Novel heterocyclic amide piperidine derivative, preparation method thereof and application thereof in hypoglycemic drugs 林剑雄 2021-08-13 CN claimed
EP-0440762-B1 5-OXY-2-PHENYLPYRIDINES AND LIQUID-CRYSTAL MATERIALS HOECHST AG (DE) 1996-07-17 EP claimed
US-5196141-A Electrooptical display MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-03-23 US claimed
EP-0440771-A1 5-OXY-2-PHENYLAZINES AND MESOMORPHOUS MEDIUM MERCK PATENT GmbH (DE) 1991-08-14 EP claimed
EP-0440762-A1 5-OXY-2-PHENYLPYRIDINES AND LIQUID-CRYSTAL MATERIALS. MERCK PATENT GMBH (DE) 1991-08-14 EP claimed
WO-1991002722-A1 5-OXY-2-PHENYLPYRIDINES AND LIQUID-CRYSTAL MATERIALS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-03-07 WO claimed
WO-1991002726-A1 5-OXY-2-PHENYLAZINES AND MESOMORPHOUS MEDIUM MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-03-07 WO claimed
US-20260078117-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS INC (US) 2026-03-19 US disclosed
US-12304907-B2 Compounds and methods of use TANGO THERAPEUTICS, INC. (US) 2025-05-20 US disclosed
US-12264154-B2 Compounds and methods of use TANGO THERAPEUTICS, INC. (US) 2025-04-01 US disclosed
CN-118994001-A NOTCH signaling pathway inhibitors and their use in cancer treatment 塞莱斯蒂亚生物技术股份公司 2024-11-22 CN disclosed
CN-113966324-B NOTCH signaling pathway inhibitors and their use in cancer treatment 塞莱斯蒂亚生物技术股份公司 2024-09-03 CN disclosed
US-20240279219-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. 2024-08-22 US disclosed
EP-0440771-A1 5-OXY-2-PHENYLAZINES AND MESOMORPHOUS MEDIUM MERCK PATENT GmbH (DE) 1991-08-14 EP disclosed
EP-0440771-A1 5-OXY-2-PHENYLAZINES AND MESOMORPHOUS MEDIUM MERCK PATENT GmbH (DE) 1991-08-14 EP disclosed
EP-0440762-A1 5-OXY-2-PHENYLPYRIDINES AND LIQUID-CRYSTAL MATERIALS. MERCK PATENT GMBH (DE) 1991-08-14 EP disclosed
WO-1991002722-A1 5-OXY-2-PHENYLPYRIDINES AND LIQUID-CRYSTAL MATERIALS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-03-07 WO disclosed
WO-1991002722-A1 5-OXY-2-PHENYLPYRIDINES AND LIQUID-CRYSTAL MATERIALS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-03-07 WO disclosed
WO-1991002726-A1 5-OXY-2-PHENYLAZINES AND MESOMORPHOUS MEDIUM MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-03-07 WO disclosed
WO-1991002726-A1 5-OXY-2-PHENYLAZINES AND MESOMORPHOUS MEDIUM MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-03-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240279219-A1 COMPOUNDS AND METHODS OF USE F12, C1R, ABCG2 LDHA 2432/4885CYP11B1 68/4885CYP11B2 86/4885
US-12264154-B2 Compounds and methods of use F12, C1R, ABCG2 LDHA 2432/4885CYP11B1 68/4885CYP11B2 86/4885
US-12304907-B2 Compounds and methods of use F12, C1R, ABCG2 LDHA 2432/4885CYP11B1 68/4885CYP11B2 86/4885
US-20260078117-A1 COMPOUNDS AND METHODS OF USE NR3C2, ADRA1A, CNR1 LDHA 1056/4885CYP11B1 104/4885CYP11B2 92/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.