SCHEMBL8519336

SCHEMBL8519336

CCCCCSc1ccccc1C#N

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.48
AR P10275 3/20 0.46
TSHR P16473 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 1/20 0.44
GAA P10253 1/20 0.44
HTT P42858 1/20 0.44
HSD17B10 Q99714 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
CYSLTR2 Q9NS75 1/20 0.42
CYSLTR1 Q9Y271 1/20 0.42
MAPT P10636 1/20 0.40
THRB P10828 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5983793 0.98 PTGS2 (0.49) PTGS2ARTSHRMEN1KMT2A
SCHEMBL2980868 0.98 PTGS2 (0.49) PTGS2ARTSHRMEN1KMT2A
SCHEMBL8400694 0.95 AR (0.50) PTGS2ARTSHRMEN1KMT2A
SCHEMBL29601087 0.95 AR (0.50) PTGS2ARTSHRMEN1KMT2A
SCHEMBL6230783 0.87 AR (0.47) PTGS2ARTSHRKDM4EGAA
SCHEMBL27613330 0.85 MEN1 (0.42) PTGS2ARTSHRMEN1KMT2A
SCHEMBL9644566 0.84 MEN1 (0.44) PTGS2ARTSHRMEN1KMT2A
SCHEMBL7713273 0.84 MEN1 (0.44) PTGS2ARTSHRMEN1KMT2A
SCHEMBL28524164 0.84 MEN1 (0.44) PTGS2ARTSHRMEN1KMT2A
SCHEMBL27652067 0.80 AR (0.44) PTGS2ARTSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111217731-B Ortho-imine ester or cyano-substituted aryl thioether derivative, preparation and application thereof 广东工业大学 2022-06-03 CN disclosed
CN-111217731-A Ortho-imine ester or cyano-substituted aryl thioether derivative, preparation and application thereof 广东工业大学 2020-06-02 CN disclosed
EP-0748311-B1 THERAPEUTIC BENZONITRILES WELLCOME FOUND (GB) 1999-08-04 EP disclosed
EP-0748311-B1 THERAPEUTIC BENZONITRILES WELLCOME FOUND (GB) 1999-08-04 EP disclosed
US-5723452-A Therapeutic benzonitriles GLAXO WELLCOME INC. (US) 1998-03-03 US disclosed
EP-0748311-A1 THERAPEUTIC BENZONITRILES THE WELLCOME FOUNDATION LIMITED (GB) 1996-12-18 EP disclosed
EP-0748311-A1 THERAPEUTIC BENZONITRILES THE WELLCOME FOUNDATION LIMITED (GB) 1996-12-18 EP disclosed
EP-0746542-A1 THERAPEUTIC BENZONITRILES THE WELLCOME FOUNDATION LIMITED (GB) 1996-12-11 EP disclosed
EP-0746542-A1 THERAPEUTIC BENZONITRILES THE WELLCOME FOUNDATION LIMITED (GB) 1996-12-11 EP disclosed
WO-1995023134-A1 THERAPEUTIC BENZONITRILES THE WELLCOME FOUNDATION LIMITED (GB) 1995-08-31 WO disclosed
WO-1995023134-A1 THERAPEUTIC BENZONITRILES THE WELLCOME FOUNDATION LIMITED (GB) 1995-08-31 WO disclosed
WO-1995023133-A1 THERAPEUTIC BENZONITRILES THE WELLCOME FOUNDATION LIMITED (GB) 1995-08-31 WO disclosed
WO-1995023133-A1 THERAPEUTIC BENZONITRILES THE WELLCOME FOUNDATION LIMITED (GB) 1995-08-31 WO disclosed