SCHEMBL29601087

SCHEMBL29601087

CCCCSc1ccccc1C#N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.50
PTGS2 P35354 6/20 0.47
MAPT P10636 2/20 0.44
THRB P10828 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
TSHR P16473 4/20 0.42
TLR8 Q9NR97 1/20 0.42
ALDH1A1 P00352 3/20 0.40
HSD17B10 Q99714 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
ALOX15 P16050 1/20 0.40
MAPK1 P28482 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8400694 1.00 AR (0.50) ARPTGS2MAPTTHRBCYP1A2
SCHEMBL8519336 0.95 PTGS2 (0.48) ARPTGS2MAPTTHRBCYP1A2
SCHEMBL2980868 0.93 PTGS2 (0.49) ARPTGS2CYP1A2CYP3A4CYP2C9
SCHEMBL5983793 0.93 PTGS2 (0.49) ARPTGS2CYP1A2CYP3A4CYP2C9
SCHEMBL6230783 0.89 AR (0.47) ARPTGS2MAPTCYP1A2CYP3A4
SCHEMBL27652067 0.85 AR (0.44) ARPTGS2MAPTTHRBTSHR
SCHEMBL28024924 0.83 AR (0.52) ARPTGS2MAPTTHRBTSHR
SCHEMBL4599675 0.81 AR (0.50) ARMAPTCYP1A2CYP3A4CYP2C9
SCHEMBL8672850 0.80 PTGS2 (0.59) PTGS2MAPTTLR8ALDH1A1L3MBTL1
SCHEMBL27613330 0.80 MEN1 (0.42) ARPTGS2MAPTTHRBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4237407-A1 PROCESS FOR PREPARING 1,2-BENZISOTHIAZOLINE-3-ONE THOR GmbH (DE) 2023-09-06 EP disclosed
CN-116457337-A Method for preparing 1, 2-benzisothiazolin-3-one 托尔有限公司 2023-07-18 CN disclosed
WO-2022089774-A1 PROCESS FOR PREPARING 1,2-BENZISOTHIAZOLINE-3-ONE THOR GMBH (DE) 2022-05-05 WO disclosed