SCHEMBL8519908

SCHEMBL8519908

Cc1cccc2c1NC(=O)C=NC2C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CREBBP Q92793 2/20 0.38
DAO P14920 1/20 0.38
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA12 O43570 1/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
HTR5A P47898 3/20 0.34
HTR2C P28335 3/20 0.34
HTR1A P08908 2/20 0.34
HTR1D P28221 2/20 0.34
HTR7 P34969 2/20 0.34
POLB P06746 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
PDK2 Q15119 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24112230 0.70 ALDH1A1 (0.43) ALDH1A1MEN1KMT2ACREBBPDAO
SCHEMBL24112725 0.70 ALDH1A1 (0.43) ALDH1A1MEN1KMT2ACREBBPDAO
SCHEMBL11368666 0.63 ALDH1A1 (0.43) ALDH1A1MEN1KMT2ACREBBPDAO
SCHEMBL24029075 0.63 TP53 (0.40) ALDH1A1MEN1KMT2ACREBBPDAO
SCHEMBL2987129 0.63 ALDH1A1 (0.44) ALDH1A1MEN1KMT2ACREBBPDAO
SCHEMBL24019657 0.63 TP53 (0.40) ALDH1A1MEN1KMT2ACREBBPDAO
SCHEMBL11368672 0.63 DAO (0.40) ALDH1A1MEN1KMT2ACREBBPDAO
SCHEMBL4474244 0.61 HTR2C (0.49) ALDH1A1MEN1KMT2ACREBBPDAO
SCHEMBL13627318 0.61 HTR2C (0.49) ALDH1A1MEN1KMT2ACREBBPDAO
SCHEMBL4476708 0.61 HTR2C (0.49) ALDH1A1MEN1KMT2ACREBBPDAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934282-A1 1,4-BENZODIAZEPINONES AND THEIR USES AS CCK ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-08-11 EP disclosed
WO-1998015535-A1 1,4-BENZODIAZEPINONES AND THEIR USES AS CCK ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-04-16 WO disclosed