SCHEMBL8520160

SCHEMBL8520160

Cc1cccc2c1N(NC(=O)OCc1ccccc1)C(=O)CN=C2CO

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.37
TNKS O95271 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
CASP3 P42574 1/20 0.36
BRD4 O60885 3/20 0.36
BRD2 P25440 3/20 0.36
BRD3 Q15059 3/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
POLB P06746 1/20 0.35
PTPN1 P18031 1/20 0.35
EPHX1 P07099 1/20 0.35
CASP1 P29466 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7828642 0.75 HDAC3 (0.51) RAB9AL3MBTL1SMN1; SMN2BRD4BRD2
SCHEMBL8542158 0.71 CYP3A4 (0.39) SMN1; SMN2BRD4BRD2BRD3CYP3A4
SCHEMBL5638173 0.70 MEN1 (0.60) RAB9ANPC1L3MBTL1SMN1; SMN2CASP3
SCHEMBL8553126 0.70 MEN1 (0.42) RAB9ANPC1SMN1; SMN2POLBNPSR1
SCHEMBL8547679 0.69 GRIN2B (0.38) L3MBTL1BRD4BRD2BRD3CYP3A4
SCHEMBL876242 0.68 CASP1 (0.48) RAB9ANPC1SMN1; SMN2POLBCASP1
Carbamic Acid SCHEMBL29087081 0.67 MEN1 (0.56) RAB9ANPC1L3MBTL1SMN1; SMN2CASP3
SCHEMBL7543329 0.65 SENP1 (0.51) RAB9ANPC1BRD4BRD2BRD3
SCHEMBL7544354 0.65 SENP1 (0.51) RAB9ANPC1BRD4BRD2BRD3
SCHEMBL7544783 0.65 SCN9A (0.51) RAB9ANPC1BRD4BRD2BRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934282-A1 1,4-BENZODIAZEPINONES AND THEIR USES AS CCK ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-08-11 EP disclosed
WO-1998015535-A1 1,4-BENZODIAZEPINONES AND THEIR USES AS CCK ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-04-16 WO disclosed