SCHEMBL8522145

SCHEMBL8522145

NC(=O)CCC1CC(c2ccc(C3=CCN(C4=NC(=O)CS4)CC3)cc2)=NO1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ITGB3 P05106 8/20 0.36
ITGA2B P08514 8/20 0.36
MIF P14174 10/20 0.35
HDAC6 Q9UBN7 1/20 0.34
ITGB2 P05107 1/20 0.33
ITGAM P11215 1/20 0.33
F2 P00734 1/20 0.33
F10 P00742 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7508461 0.83 MIF (0.38) NPC1RAB9AMIFHDAC6
SCHEMBL7502963 0.74 MIF (0.40) MIF
SCHEMBL7502407 0.73 MIF (0.35) RAB9AMIF
SCHEMBL7505315 0.67 MIF (0.38) NPC1RAB9AMIFHDAC6
SCHEMBL7505771 0.63 MIF (0.38) NPC1RAB9AMIFHDAC6
SCHEMBL14350426 0.62 QDPR (0.49) MIFHDAC6
SCHEMBL7507435 0.62 MIF (0.42) RAB9AMIF
SCHEMBL7504359 0.61 QDPR (0.46) NPC1RAB9AMIFHDAC6
SCHEMBL7505583 0.61 RAB9A (0.45) NPC1RAB9AMIFHDAC6
SCHEMBL12556312 0.60 MIF (0.74) NPC1RAB9AITGB3ITGA2BMIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0920421-A1 ISOXAZOLINE DERIVATIVES USEFUL AS ANTIMICROBIALS PHARMACIA & UPJOHN COMPANY (US) 1999-06-09 EP claimed
WO-1998007708-A1 ISOXAZOLINE DERIVATIVES USEFUL AS ANTIMICROBIALS PHARMACIA & UPJOHN COMPANY (US) 1998-02-26 WO claimed