SCHEMBL8522611

SCHEMBL8522611

COc1ccc(NC(C)=O)c(OCCCCl)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
HSD17B1 P14061 1/20 0.54
HSD17B2 P37059 1/20 0.54
MAPT P10636 4/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
PKM P14618 1/20 0.51
HPGD P15428 2/20 0.50
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
BRD4 O60885 1/20 0.48
PTK2 Q05397 1/20 0.48
CYP1A1 P04798 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP1B1 Q16678 1/20 0.48
LMNA P02545 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2795656 0.88 ALDH1A1 (0.54) ALDH1A1HSD17B1HSD17B2MAPTMEN1
SCHEMBL30622065 0.82 HSD17B1 (0.75) ALDH1A1HSD17B1HSD17B2MAPTMEN1
SCHEMBL2191052 0.82 HSD17B1 (0.75) ALDH1A1HSD17B1HSD17B2MAPTMEN1
SCHEMBL3959073 0.80 FLT3 (0.54) ALDH1A1HSD17B1HSD17B2MAPTMEN1
SCHEMBL3860865 0.80 ALDH1A1 (0.54) ALDH1A1HSD17B1HSD17B2MAPTMEN1
SCHEMBL7789182 0.78 LMNA (0.50) LMNASMN1; SMN2
SCHEMBL5718254 0.77 CYP19A1 (0.67) ALDH1A1MAPTMEN1KMT2APKM
SCHEMBL4216922 0.77 ALDH1A1 (0.51) ALDH1A1HSD17B1HSD17B2MAPTMEN1
SCHEMBL4216929 0.77 ALDH1A1 (0.51) ALDH1A1HSD17B1HSD17B2MAPTMEN1
SCHEMBL10600631 0.77 HTT (0.48) ALDH1A1HSD17B1HSD17B2MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0957102-A1 Heteroarylpiperidines and piperazines and their use as antipsychotics and analgetics HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1999-11-17 EP disclosed