SCHEMBL8523648

SCHEMBL8523648

CCCCCC1CNc2ccccc21

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.47
CCKBR P32239 2/20 0.38
CYSLTR2 Q9NS75 1/20 0.37
CYSLTR1 Q9Y271 1/20 0.37
HTR5A P47898 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28756698 0.98 BCHE (0.46) BCHECCKBRCYSLTR2CYSLTR1
SCHEMBL22582292 0.98 BCHE (0.46) BCHECCKBRCYSLTR2CYSLTR1
SCHEMBL7074697 0.95 BCHE (0.48) BCHECCKBRHTR5A
SCHEMBL8261364 0.88 HTR5A (0.41) BCHECCKBRHTR5A
SCHEMBL1325640 0.85 SIGMAR1 (0.42) BCHECCKBR
SCHEMBL7692638 0.84 BCHE (0.64) BCHECYSLTR2CYSLTR1HTR5A
Dimethylamine SCHEMBL8649623 0.83 BCHE (0.39) BCHECCKBRHTR5A
SCHEMBL5546413 0.83 CCKBR (0.38) BCHECCKBR
SCHEMBL20879359 0.82 BCHE (0.37) BCHECCKBR
SCHEMBL5542142 0.82 CCKBR (0.37) BCHECCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101255170-A 2,3-dihydroimidazo[2,1-b]oxazole compound OTSUKA PHARMA CO LTD (JP) 2008-09-03 CN disclosed
CN-101172981-A 2,3-dihydroimidazo[2,1-b]oxazole compound OTSUKA PHARMA CO LTD (JP) 2008-05-07 CN disclosed
CN-100366624-C 2, 3-dihydro-6-nitroimidazo [2,1-b ] * azole compounds OTSUKA PHARMA CO LTD (JP) 2008-02-06 CN disclosed
CN-1705670-A 2, 3-dihydro-6-nitroimidazo [2, 1-b ] oxazole compounds OTSUKA PHARMA CO LTD (JP) 2005-12-07 CN disclosed
US-5936098-A Process for producing indoline compounds and intermediates for the production of the same TOKYO TANABE COMPANY LIMITED (JP) 1999-08-10 US disclosed
US-5936098-A Process for producing indoline compounds and intermediates for the production of the same TOKYO TANABE COMPANY LIMITED (JP) 1999-08-10 US disclosed
EP-0810214-A4 PROCESS FOR PRODUCING INDOLINE COMPOUNDS AND INTERMEDIATES FOR THE PRODUCTION OF THE SAME TOKYO TANABE CO (JP) 1998-06-10 EP disclosed
EP-0810214-A1 PROCESS FOR PRODUCING INDOLINE COMPOUNDS AND INTERMEDIATES FOR THE PRODUCTION OF THE SAME TOKYO TANABE COMPANY LIMITED (JP) 1997-12-03 EP disclosed
EP-0810214-A1 PROCESS FOR PRODUCING INDOLINE COMPOUNDS AND INTERMEDIATES FOR THE PRODUCTION OF THE SAME TOKYO TANABE COMPANY LIMITED (JP) 1997-12-03 EP disclosed
WO-1996025396-A1 PROCESS FOR PRODUCING INDOLINE COMPOUNDS AND INTERMEDIATES FOR THE PRODUCTION OF THE SAME TOKYO TANABE COMPANY LIMITED (JP) 1996-08-22 WO disclosed
US-4153789-A HYPOGLYCEMIC AGENTS, ANTICOAGULANTS DELMAR CHEMICALS LIMITED (CA) 1979-05-08 US disclosed
US-4080330-A HYPOGLYCEMIC AGENTS, ANTICOAGULANTS DELMAR CHEMICALS LIMITED (CA) 1978-03-21 US disclosed