SCHEMBL8523769

SCHEMBL8523769

CCN(CC)CC(=O)Nc1c2c(nc3ccccc13)CCCC2

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.62
BCHE P06276 2/20 0.61
HTT P42858 2/20 0.60
GAA P10253 1/20 0.60
ACHE P22303 1/20 0.59
MEN1 O00255 1/20 0.58
USP2 O75604 1/20 0.58
ALDH1A1 P00352 1/20 0.58
KMT2A Q03164 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
CACNA2D1 P54289 1/20 0.57
APP P05067 3/20 0.57
MAPT P10636 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9232310 0.88 KDM4E (0.64) KDM4EBCHEHTTGAAACHE
SCHEMBL9748781 0.87 KDM4E (0.68) KDM4EBCHEHTTGAAACHE
SCHEMBL9387187 0.86 KDM4E (0.69) KDM4EBCHEHTTGAAACHE
SCHEMBL8474173 0.83 BCHE (0.66) KDM4EBCHEHTTGAAACHE
SCHEMBL9747358 0.83 KDM4E (0.63) KDM4EBCHEHTTGAAACHE
SCHEMBL9384234 0.82 KDM4E (0.72) KDM4EBCHEHTTGAAACHE
SCHEMBL9382159 0.82 KDM4E (0.65) KDM4EBCHEHTTGAAACHE
SCHEMBL27524922 0.81 BCHE (0.63) KDM4EBCHEHTTGAAACHE
SCHEMBL13624997 0.81 KDM4E (0.61) KDM4EBCHEHTTGAAACHE
SCHEMBL9748588 0.81 KDM4E (0.66) KDM4EBCHEHTTGAAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861411-A TREATING DISTURBANCES OF MEMORY SUCH AS SENILE DEMENTIA AND ALZHEIMER'S DISEASE MITSUBISHI CHEMICAL CORPORATION (JP) 1999-01-19 US disclosed
US-5536728-A TREATMENT OF SENILE DEMENTIA AND ALZHEIMER'S DISEASE MITSUBISHI CHEMICAL CORPORATION (JP) 1996-07-16 US disclosed
EP-0427636-B1 4-Acylaminopyridine derivatives MITSUBISHI CHEM CORP (JP) 1996-05-29 EP disclosed
US-5397785-A Activators of cholinergic neurons to treat memory disorders such as senile dementia and Alzheimer's disease MITSUBISHI KASEI CORPORATION (JP) 1995-03-14 US disclosed
EP-0319429-B1 9-Acylamino-tetrahydroacridine derivatives and memory enhancing agent containing said derivative as active ingredient MITSUBISHI CHEM IND (JP) 1994-04-27 EP disclosed
EP-0427636-A2 4-Acylaminopyridine derivatives Mitsubishi Chemical Corporation (JP) 1991-05-15 EP disclosed
US-4985430-A ALZHEIMER*S DISEASE MITSUBISHI KASEI CORPORATION (JP) 1991-01-15 US disclosed
EP-0319429-A2 9-Acylamino-tetrahydroacridine derivatives and memory enhancing agent containing said derivative as active ingredient MITSUBISHI KASEI CORPORATION (JP) 1989-06-07 EP disclosed