SCHEMBL8523935

SCHEMBL8523935

Cc1cc2c(cc1-c1csc(-c3ccncc3)n1)CCCC(=O)N2

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MAPT P10636 2/20 0.44
MMP12 P39900 1/20 0.44
CDK5 Q00535 13/20 0.43
CDK5R1 Q15078 13/20 0.43
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
HTT P42858 1/20 0.40
CYP19A1 P11511 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8525368 0.82 SMN1; SMN2 (0.60) NPC1RAB9AMAPTMMP12CDK5
SCHEMBL8523719 0.82 CDK5 (0.44) NPC1RAB9AMAPTMMP12CDK5
SCHEMBL8525110 0.81 CDK5 (0.42) NPC1RAB9AMAPTMMP12CDK5
SCHEMBL8525334 0.76 CDK5 (0.39) NPC1RAB9ACDK5CDK5R1SMN1; SMN2
SCHEMBL8525270 0.75 SMN1; SMN2 (0.70) NPC1RAB9AMAPTMMP12CDK5
SCHEMBL6651931 0.72 MAPT (0.65) NPC1RAB9AMAPTMMP12CDK5
SCHEMBL6394131 0.70 PDE3B (0.61) PDE3BPDE3ACYP19A1
SCHEMBL8480061 0.69 PDE3B (0.68) NPC1RAB9AMAPTMMP12CDK5
SCHEMBL23657751 0.69 CYP17A1 (0.73) NPC1RAB9AMAPTCDK5CDK5R1
SCHEMBL8484612 0.68 RAB9A (0.47) NPC1RAB9AMAPTMMP12CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999015524-A1 THIAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-04-01 WO disclosed