SCHEMBL8525110

SCHEMBL8525110

Cc1cc2c(cc1-c1csc(-c3ccncc3)n1)C(C)(C)CCC(=O)N2

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 13/20 0.42
CDK5R1 Q15078 13/20 0.42
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
KDM4E B2RXH2 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP19A1 P11511 1/20 0.38
MAPT P10636 1/20 0.38
MMP12 P39900 1/20 0.38
CYP17A1 P05093 1/20 0.38
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8523935 0.81 NPC1 (0.44) CDK5CDK5R1NPC1RAB9AKDM4E
SCHEMBL8524244 0.78 CDK5 (0.38) CDK5CDK5R1NPC1RAB9AKDM4E
SCHEMBL8524612 0.75 CYP19A1 (0.54) NPC1RAB9AKDM4ESMN1; SMN2CYP19A1
SCHEMBL8523719 0.74 CDK5 (0.44) CDK5CDK5R1NPC1RAB9AKDM4E
SCHEMBL8523780 0.73 CYP19A1 (0.48) CDK5CDK5R1NPC1RAB9AKDM4E
SCHEMBL8524764 0.71 CYP19A1 (0.45) CDK5CDK5R1NPC1RAB9AKDM4E
SCHEMBL8525270 0.69 SMN1; SMN2 (0.70) CDK5CDK5R1NPC1RAB9AKDM4E
SCHEMBL8524322 0.69 CDC25A (0.49) CDK5CDK5R1NPC1RAB9AKDM4E
SCHEMBL8525368 0.68 SMN1; SMN2 (0.60) CDK5CDK5R1NPC1RAB9AKDM4E
SCHEMBL23657751 0.67 CYP17A1 (0.73) CDK5CDK5R1NPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999015524-A1 THIAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-04-01 WO disclosed