SCHEMBL8525447

SCHEMBL8525447

N#Cc1ccc(CNC(=O)c2cccc3cc(NS(=O)(=O)c4cccc5scnc45)ccc23)cc1

nearest known ligand 0.44

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PKLR P30613 18/20 0.44
MCL1 Q07820 1/20 0.38
CNR2 P34972 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8525044 0.87 PKLR (0.49) PKLR
SCHEMBL8524665 0.84 SLC16A3 (0.42) PKLRMCL1CNR2
SCHEMBL8524454 0.81 PKLR (0.49) PKLR
SCHEMBL1110102 0.78 TUBB (0.46) MCL1CNR2
SCHEMBL8525059 0.75 HDAC2 (0.46) CNR2
SCHEMBL8525757 0.74 KMT2A (0.44) PKLR
Hydrochloric Acid SCHEMBL8525302 0.74 F2 (0.56) PKLR
SCHEMBL8525755 0.73 HSP90AA1 (0.49) MCL1CNR2
SCHEMBL7358688 0.73 PKLR (0.47) PKLR
SCHEMBL8525436 0.71 HDAC2 (0.50) CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999029670-A2 AMINOCARBONYLTETRALIN AND DIHYDRONAPHTALENE DERIVATES AS THROMBIN INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-17 WO disclosed