SCHEMBL8525757

SCHEMBL8525757

N#Cc1ccc(CNC(=O)c2cccc3cc(CCNNS(=O)(=O)c4cccc5cccnc45)ccc23)cc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.44
MEN1 O00255 1/20 0.43
EGLN1 Q9GZT9 5/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
ALDH1A1 P00352 2/20 0.39
GLO1 Q04760 1/20 0.39
PKLR P30613 1/20 0.39
NSD2 O96028 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8525044 0.86 PKLR (0.49) KMT2AMEN1EGLN1ALDH1A1GLO1
SCHEMBL8524454 0.82 PKLR (0.49) KMT2AMEN1EGLN1ALDH1A1PKLR
SCHEMBL8524665 0.77 SLC16A3 (0.42) KMT2AMEN1EGLN1ALDH1A1PKLR
SCHEMBL8489621 0.76 EGLN1 (0.46) EGLN1SMN1; SMN2ADORA2AADORA1NSD2
SCHEMBL8525447 0.74 PKLR (0.44) PKLR
SCHEMBL7358688 0.73 PKLR (0.47) KMT2AMEN1EGLN1ALDH1A1PKLR
Hydrochloric Acid SCHEMBL8525302 0.73 F2 (0.56) KMT2AMEN1ALDH1A1PKLR
SCHEMBL8525436 0.72 HDAC2 (0.50) NSD2
SCHEMBL1320296 0.72 HDAC2 (0.50) ALDH1A1NSD2
SCHEMBL8494353 0.71 HDAC2 (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999029670-A2 AMINOCARBONYLTETRALIN AND DIHYDRONAPHTALENE DERIVATES AS THROMBIN INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-17 WO disclosed